SCHEMBL4613022

SCHEMBL4613022

CCOC(=O)Oc1nc(N)sc1Br

nearest known ligand 0.45

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 9/20 0.45
CYP1A2 P05177 1/20 0.45
HPGD P15428 2/20 0.42
ALOX5 P09917 1/20 0.41
CUL4A Q13619 1/20 0.39
HSD17B10 Q99714 1/20 0.39
MAPT P10636 2/20 0.38
MEN1 O00255 1/20 0.38
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
KMT2A Q03164 1/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
GAA P10253 2/20 0.38
CA2 P00918 1/20 0.37
LMNA P02545 1/20 0.36
FBP1 P09467 1/20 0.36
POLB P06746 1/20 0.35
FHIT P49789 1/20 0.35
SOAT1 P35610 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4599801 0.81 ALDH1A1 (0.45) ALDH1A1CYP1A2HPGDALOX5CUL4A
SCHEMBL27739639 0.78 ALOX5 (0.37) ALDH1A1CYP1A2HPGDALOX5HSD17B10
SCHEMBL6931770 0.78 ALDH1A1 (0.52) ALDH1A1CYP1A2HPGDALOX5MEN1
SCHEMBL13609507 0.75 ALDH1A1 (0.53) ALDH1A1CYP1A2HPGDHSD17B10MAPT
SCHEMBL960280 0.74 ALDH1A1 (0.69) ALDH1A1CYP1A2HPGDHSD17B10MAPT
SCHEMBL9202295 0.69 ALOX5 (0.44) ALDH1A1CYP1A2HPGDALOX5CUL4A
SCHEMBL11373187 0.69 ALDH1A1 (0.46) ALDH1A1CYP1A2HPGDHSD17B10MAPT
SCHEMBL16852179 0.68 ALDH1A1 (0.39) ALDH1A1CYP1A2HPGDALOX5MAPT
SCHEMBL16852121 0.68 ALDH1A1 (0.39) ALDH1A1CYP1A2HPGDALOX5MAPT
SCHEMBL4611628 0.67 NOS1 (0.41) ALDH1A1CYP1A2HPGDHSD17B10MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1910330-B1 HETEROCYCLYLAMIDE-SUBSTITUTED THIAZOLES, PYRROLES AND THIOPHENES AICURIS GMBH & CO KG (DE) 2014-07-23 EP disclosed
EP-1910330-A1 HETEROCYCLYLAMIDE-SUBSTITUTED THIAZOLES, PYRROLES AND THIOPHENES Bayer HealthCare AG (DE) 2008-04-16 EP disclosed
WO-2007009578-A1 HETEROCYCLYLAMIDE-SUBSTITUTED THIAZOLES, PYRROLES AND THIOPHENES BAYER HEALTHCARE AG (DE) 2007-01-25 WO disclosed
EP-1371651-A2 N-alkylated Thiazoliumsalts and processes for their preparation BAYER AG (DE) 2003-12-17 EP disclosed