SCHEMBL461565

SCHEMBL461565

NC(=O)c1cnnn1Cc1c(F)cccc1F

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA5A P35218 1/20 0.51
OPRM1 P35372 1/20 0.40
OPRD1 P41143 1/20 0.40
PRMT5 O14744 1/20 0.35
KDM4E B2RXH2 3/20 0.35
PTGDR2 Q9Y5Y4 1/20 0.35
ALDH1A1 P00352 1/20 0.35
CD38 P28907 1/20 0.35
PKM P14618 3/20 0.35
CDK1 P06493 1/20 0.35
CDK4 P11802 1/20 0.35
CDK2 P24941 1/20 0.35
PKLR P30613 1/20 0.35
MAPK8 P45983 1/20 0.35
JAK2 O60674 1/20 0.34
KCNK3 O14649 1/20 0.34
HSD11B1 P28845 1/20 0.34
SLC22A12 Q96S37 1/20 0.34
KLKB1 P03952 1/20 0.34
ADORA2A P29274 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9910582 0.87 CA5A (0.43) CA5APRMT5KDM4EPTGDR2ALDH1A1
SCHEMBL10643826 0.76 CA5A (0.40) CA5AKDM4EALDH1A1PKMPKLR
SCHEMBL9857412 0.73 CA5A (0.55) CA5AOPRM1OPRD1KDM4EALDH1A1
SCHEMBL9714161 0.73 CA5A (0.48) CA5AOPRM1OPRD1KDM4EALDH1A1
SCHEMBL9476992 0.72 CA5A (0.53) CA5AALDH1A1ADORA2AADORA1
SCHEMBL10662999 0.72 LMNA (0.57) ALDH1A1
SCHEMBL16824152 0.71 CA5A (0.52) CA5AOPRM1OPRD1KDM4EPTGDR2
SCHEMBL10662727 0.71 CA5A (0.52) CA5AOPRM1OPRD1KDM4EPTGDR2
SCHEMBL30281238 0.71 HASPIN (0.36) HSD11B1
SCHEMBL22125841 0.71 MAPT (0.35) KDM4EALDH1A1HSD11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012032540-A1 PROCESS FOR PREPARATION OF FLUORINATED TRIAZOLE COMPOUND INDOCO REMEDIES LIMITED (IN) 2012-03-15 WO disclosed
WO-2012032540-A1 PROCESS FOR PREPARATION OF FLUORINATED TRIAZOLE COMPOUND INDOCO REMEDIES LIMITED (IN) 2012-03-15 WO disclosed