SCHEMBL9857412

SCHEMBL9857412

NC(=O)c1nnn(Cc2c(F)cccc2F)c1C(N)=O

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA5A P35218 1/20 0.55
ADORA2A P29274 2/20 0.39
ADORA1 P30542 2/20 0.39
ADORA3 P0DMS8 1/20 0.39
ADORA2B P29275 1/20 0.39
HPGD P15428 1/20 0.38
OPRM1 P35372 1/20 0.38
OPRD1 P41143 1/20 0.38
ALDH1A1 P00352 2/20 0.35
KDM4E B2RXH2 1/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
GALR3 O60755 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2C9 P11712 1/20 0.35
NR2F2 P24468 1/20 0.35
HIF1A Q16665 1/20 0.35
TP53 P04637 2/20 0.35
CYP1A2 P05177 1/20 0.35
MAPK8 P45983 1/20 0.35
JAK2 O60674 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9857903 0.91 CA5A (0.46) CA5AALDH1A1KDM4EMEN1TSHR
SCHEMBL10662709 0.88 CA5A (0.49) CA5AADORA2AADORA1ADORA3ADORA2B
SCHEMBL9476992 0.87 CA5A (0.53) CA5AADORA2AADORA1ADORA3ADORA2B
SCHEMBL9857464 0.86 CA5A (0.44) CA5AADORA2AADORA1ADORA3ADORA2B
SCHEMBL10662727 0.86 CA5A (0.52) CA5AADORA2AADORA1ADORA3ADORA2B
SCHEMBL9857450 0.86 GRM2 (0.45) CA5AADORA2AADORA1ADORA3ADORA2B
SCHEMBL9634851 0.79 HPGD (0.61) HPGDALDH1A1SMN1; SMN2CYP1A2MEN1
SCHEMBL9857331 0.78 TP53 (0.41) CA5AADORA2AADORA1ADORA3ADORA2B
SCHEMBL9857352 0.78 TP53 (0.43) ADORA2AADORA1ADORA3ADORA2BHPGD
SCHEMBL10670780 0.76 TP53 (0.58) CA5AALDH1A1SMN1; SMN2TP53CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0199262-B1 FLUORINATED BENZYL TRIAZOLE COMPOUNDS CIBA-GEIGY AG (CH) 1991-02-27 EP claimed
US-4789680-A Aralkyltriazole compounds CIBA-GEIGY CORPORATION (US) 1988-12-06 US claimed
EP-0199262-A2 Fluorinated benzyl triazole compounds CIBA-GEIGY AG (CH) 1986-10-29 EP claimed
EP-0199262-B1 FLUORINATED BENZYL TRIAZOLE COMPOUNDS CIBA-GEIGY AG (CH) 1991-02-27 EP disclosed
US-4789680-A Aralkyltriazole compounds CIBA-GEIGY CORPORATION (US) 1988-12-06 US disclosed
EP-0199262-A2 Fluorinated benzyl triazole compounds CIBA-GEIGY AG (CH) 1986-10-29 EP disclosed