SCHEMBL4615976

SCHEMBL4615976

O=S(=O)(NCc1ccc(Cl)nc1)c1cc(S(=O)(=O)c2ccccc2)ccc1C(F)(F)F

nearest known ligand 0.55

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
SFRP1 Q8N474 13/20 0.55
CYP2C9 P11712 1/20 0.51
NAMPT P43490 1/20 0.51
MEN1 O00255 1/20 0.50
KMT2A Q03164 1/20 0.50
CYP2C19 P33261 1/20 0.49
ALDH1A1 P00352 2/20 0.48
PKM P14618 1/20 0.48
WNT3 P56703 3/20 0.48
GAA P10253 1/20 0.46
LMNA P02545 2/20 0.45
SLC12A2 P55011 1/20 0.45
SLC12A5 Q9H2X9 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4637732 0.91 CYP2C9 (0.48) SFRP1CYP2C9NAMPTMEN1KMT2A
SCHEMBL4637735 0.86 CYP2C9 (0.49) SFRP1CYP2C9NAMPTMEN1KMT2A
SCHEMBL6101796 0.84 SFRP1 (0.60) SFRP1WNT3
SCHEMBL4617728 0.82 LMNA (0.60) SFRP1NAMPTWNT3LMNA
SCHEMBL4616485 0.82 SFRP1 (0.52) SFRP1WNT3LMNASLC12A2SLC12A5
SCHEMBL4617999 0.82 SFRP1 (0.52) SFRP1WNT3LMNASLC12A2SLC12A5
SCHEMBL4637484 0.81 SFRP1 (0.62) SFRP1NAMPTALDH1A1WNT3
SCHEMBL4618553 0.80 SFRP1 (0.59) SFRP1WNT3
SCHEMBL4617769 0.79 SFRP1 (0.56) SFRP1PKMWNT3GAALMNA
SCHEMBL4616901 0.78 SFRP1 (0.50) SFRP1WNT3LMNASLC12A2SLC12A5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101208299-A Diarylsulfone sulfonamides and use therof WYETH CORP (US) 2008-06-25 CN claimed
EP-1879859-A2 DIARYLSULFONE SULFONAMIDES AND USE THEROF Wyeth a Corporation of the State of Delaware (US) 2008-01-23 EP claimed
US-20060276464-A1 Diarylsulfone sulfonamides and use thereof WYETH (US) 2006-12-07 US claimed
WO-2006124875-A2 DIARYLSULFONE SULFONAMIDES AND USE THEROF WYETH (US) 2006-11-23 WO claimed
CN-101208299-A Diarylsulfone sulfonamides and use therof WYETH CORP (US) 2008-06-25 CN disclosed
EP-1879859-A2 DIARYLSULFONE SULFONAMIDES AND USE THEROF Wyeth a Corporation of the State of Delaware (US) 2008-01-23 EP disclosed
US-20060276464-A1 Diarylsulfone sulfonamides and use thereof WYETH (US) 2006-12-07 US disclosed
WO-2006124875-A2 DIARYLSULFONE SULFONAMIDES AND USE THEROF WYETH (US) 2006-11-23 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060276464-A1 Diarylsulfone sulfonamides and use thereof SFRP1, SOS1, FZD7 SFRP1 1/4885CYP2C9 1693/4885NAMPT 3852/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.