SCHEMBL4617633

SCHEMBL4617633

CCCC(=O)OOc1ccc(C(=C2CC(C)(C)CC(C)(C)C2)c2ccc(F)cc2)cc1

nearest known ligand 0.35

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HTR7 P34969 1/20 0.35
OPRD1 P41143 2/20 0.35
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
SLC6A2 P23975 1/20 0.32
SLC6A3 Q01959 1/20 0.32
MAOB P27338 2/20 0.32
BCL9 O00512 1/20 0.32
CTNNB1 P35222 1/20 0.32
ESR1 P03372 1/20 0.32
RXRA P19793 2/20 0.31
PLA2G7 Q13093 1/20 0.31
CYP2C9 P11712 1/20 0.31
TSHR P16473 1/20 0.31
GAA P10253 2/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
OPRM1 P35372 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4617631 0.88 BCL9 (0.44) HTR7OPRD1RAB9ASLC6A2SLC6A3
SCHEMBL3135615 0.84 ESR1 (0.39) OPRD1NPC1RAB9ASLC6A2SLC6A3
SCHEMBL3562321 0.77 SMN1; SMN2 (0.46) OPRD1
SCHEMBL3087766 0.77 HRH2 (0.44) MAOBL3MBTL1
SCHEMBL3135618 0.77 ESR1 (0.54) OPRD1SLC6A2SLC6A3MAOBESR1
SCHEMBL3069744 0.76 LMNA (0.42) MAOBGAAL3MBTL1
SCHEMBL3075680 0.76 LTA4H (0.46) PLA2G7L3MBTL1
SCHEMBL3074106 0.75 BCL2L1 (0.49) HTR7OPRD1ESR1RXRATSHR
SCHEMBL4728801 0.74 FFAR4 (0.34) OPRD1SLC6A2SLC6A3PLA2G7CYP2C9
SCHEMBL3082749 0.73 NR1I2 (0.43) MAOBESR1PLA2G7GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1891026-A2 CYCLOALKYLIDENE COMPOUNDS AS SELECTIVE ESTROGEN RECEPTOR MODULATORS Smithkline Beecham Corporation (US) 2008-02-27 EP disclosed
WO-2006127871-A2 CYCLOALKYLIDENE COMPOUNDS AS SELECTIVE ESTROGEN RECEPTOR MODULATORS SMITHKLINE BEECHAM CORPORATION (US) 2006-11-30 WO disclosed