SCHEMBL46199

SCHEMBL46199

COC/C(=C/c1ccc(-c2ccc(C(=O)O)cc2)o1)SC(=O)NCc1ccc(F)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
XPA P23025 3/20 0.48
KDM4E B2RXH2 5/20 0.47
ALDH1A1 P00352 3/20 0.47
LMNA P02545 1/20 0.47
HPGD P15428 1/20 0.47
POLB P06746 5/20 0.46
TDP1 Q9NUW8 4/20 0.46
MEN1 O00255 3/20 0.46
KMT2A Q03164 3/20 0.46
L3MBTL1 Q9Y468 2/20 0.46
NPC1 O15118 2/20 0.46
RAB9A P51151 2/20 0.46
ENPP2 Q13822 1/20 0.45
MAPT P10636 2/20 0.44
PKM P14618 1/20 0.44
PHGDH O43175 2/20 0.44
PTPN1 P18031 1/20 0.39
KEAP1 Q14145 1/20 0.39
NFE2L2 Q16236 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL46709 0.83 XPA (0.51) XPAKDM4EALDH1A1LMNAHPGD
SCHEMBL27941201 0.64 KMT2A (0.62) ALDH1A1LMNAHPGDKMT2A
SCHEMBL16346518 0.64 HPGD (0.53) KDM4EALDH1A1HPGDPOLBTDP1
SCHEMBL3057812 0.64 HPGD (0.69) KDM4EALDH1A1LMNAHPGDNPC1
SCHEMBL3054179 0.64 ALDH1A1 (0.70) KDM4EALDH1A1LMNAHPGDMEN1
SCHEMBL23135764 0.63 GAA (0.68) ALDH1A1LMNAHPGDMEN1KMT2A
SCHEMBL10099566 0.63 NR1H4 (0.69) LMNAKMT2AL3MBTL1
SCHEMBL4946307 0.63 LMNA (0.57) KDM4EALDH1A1LMNAHPGDPOLB
Fluorobenzene SCHEMBL27605534 0.62 KMT2A (0.55) KDM4EALDH1A1LMNAHPGDPOLB
SCHEMBL684546 0.62 ENPP2 (1.00) KDM4EALDH1A1LMNAHPGDPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012005800-A1 COMPOUNDS AND METHODS FOR REGULATING INTEGRIN CD11B/CD18 ADHAERE PHARAMACEUTICALS, INC. (US) 2012-01-12 WO disclosed