SCHEMBL4621072

SCHEMBL4621072

NC(=O)[C@H](CCC(=O)O)N(CCCc1ccccc1)C(=O)c1ccc2c(c1)C(=O)c1ccccc1-2

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.40
MAPT P10636 2/20 0.40
NPC1 O15118 1/20 0.40
ALDH1A1 P00352 1/20 0.40
LMNA P02545 1/20 0.40
RAB9A P51151 1/20 0.40
HTR7 P34969 1/20 0.40
HTR2B P41595 1/20 0.40
TTR P02766 1/20 0.40
PTPRC P08575 4/20 0.39
CTSL P07711 1/20 0.38
PTPN13 Q12923 1/20 0.38
HDAC3 O15379 1/20 0.36
MAPK1 P28482 1/20 0.36
ADRA1A P35348 1/20 0.36
HDAC4 P56524 1/20 0.36
SLC6A3 Q01959 1/20 0.36
HDAC1 Q13547 1/20 0.36
HDAC7 Q8WUI4 1/20 0.36
HDAC2 Q92769 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4621074 0.88 NPC1 (0.40) SMN1; SMN2MAPTNPC1ALDH1A1LMNA
SCHEMBL2246521 0.88 HTR7 (0.40) SMN1; SMN2MAPTNPC1ALDH1A1LMNA
SCHEMBL4623203 0.88 NPC1 (0.43) SMN1; SMN2MAPTNPC1ALDH1A1LMNA
SCHEMBL4622938 0.87 HTR7 (0.39) SMN1; SMN2MAPTNPC1ALDH1A1LMNA
SCHEMBL5653519 0.85 CYP1A2 (0.44) SMN1; SMN2MAPTHDAC3MAPK1ADRA1A
SCHEMBL2248130 0.82 TAS2R14 (0.39) SMN1; SMN2MAPTNPC1ALDH1A1LMNA
SCHEMBL5653109 0.81 SRD5A2 (0.47) LPAR1PTGDR2MMP2
SCHEMBL5651545 0.80 MMP12 (0.44) SMN1; SMN2MAPTALDH1A1LMNARAB9A
SCHEMBL2244942 0.75 NPC1 (0.42) SMN1; SMN2MAPTNPC1ALDH1A1LMNA
SCHEMBL4623232 0.73 HTR7 (0.38) SMN1; SMN2MAPTNPC1ALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1902014-A2 GLUTAMATE AGGRECANASE INHIBITORS Wyeth (US) 2008-03-26 EP disclosed
WO-2007008994-A2 GLUTAMATE AGGRECANASE INHIBITORS WYETH (US) 2007-01-18 WO disclosed