SCHEMBL4621074

SCHEMBL4621074

NC(=O)CC[C@@H](C(=O)O)N(CCCc1ccccc1)C(=O)c1ccc2c(c1)C(=O)c1ccccc1-2

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.40
RAB9A P51151 3/20 0.40
MAPT P10636 2/20 0.40
ALDH1A1 P00352 2/20 0.40
LMNA P02545 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
HTR7 P34969 1/20 0.40
HTR2B P41595 1/20 0.40
TTR P02766 1/20 0.40
PTPRC P08575 4/20 0.39
GRIK1 P39086 1/20 0.37
CTSL P07711 1/20 0.36
PTPN13 Q12923 1/20 0.36
LPAR1 Q92633 2/20 0.36
ACHE P22303 1/20 0.35
ALOX5 P09917 1/20 0.34
ATM Q13315 1/20 0.34
GRIN1 Q05586 1/20 0.34
GRIN2A Q12879 1/20 0.34
GRIN2B Q13224 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4621072 0.88 SMN1; SMN2 (0.40) NPC1RAB9AMAPTALDH1A1LMNA
SCHEMBL2246521 0.76 HTR7 (0.40) NPC1RAB9AMAPTALDH1A1LMNA
SCHEMBL4622938 0.75 HTR7 (0.39) NPC1RAB9AMAPTALDH1A1LMNA
SCHEMBL4623203 0.75 NPC1 (0.43) NPC1RAB9AMAPTALDH1A1LMNA
SCHEMBL5653519 0.72 CYP1A2 (0.44) MAPTSMN1; SMN2KDM4ECYP1A2
SCHEMBL2248130 0.70 TAS2R14 (0.39) NPC1RAB9AMAPTALDH1A1LMNA
SCHEMBL4371351 0.69 KMT2A (0.40) ALDH1A1LMNASMN1; SMN2KDM4EL3MBTL1
SCHEMBL2249427 0.69 CA2 (0.59) NPC1RAB9AMAPTALDH1A1HTR7
SCHEMBL5653109 0.68 SRD5A2 (0.47) LPAR1
SCHEMBL4621965 0.68 TRIM24 (0.37) MAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1902014-A2 GLUTAMATE AGGRECANASE INHIBITORS Wyeth (US) 2008-03-26 EP disclosed
WO-2007008994-A2 GLUTAMATE AGGRECANASE INHIBITORS WYETH (US) 2007-01-18 WO disclosed