SCHEMBL4622159

SCHEMBL4622159

COC(=O)C=Cc1ccc(N2CCCCC2)nc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.47
CA1 P00915 1/20 0.47
CA2 P00918 1/20 0.47
TYR P14679 1/20 0.47
CA7 P43166 1/20 0.47
CA9 Q16790 1/20 0.47
CA14 Q9ULX7 1/20 0.47
SMN1; SMN2 Q16637 3/20 0.46
KDM4E B2RXH2 2/20 0.46
KMT2A Q03164 2/20 0.46
AOC3 Q16853 2/20 0.44
FDPS P14324 1/20 0.44
TTR P02766 1/20 0.43
APP P05067 1/20 0.43
TRPV1 Q8NER1 1/20 0.42
ALDH1A1 P00352 4/20 0.42
NPSR1 Q6W5P4 2/20 0.42
LMNA P02545 1/20 0.42
MAPT P10636 1/20 0.42
ALOX12 P18054 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3784306 0.87 ALDH1A1 (0.49) CA12CA1CA2TYRCA7
SCHEMBL3683824 0.87 CA12 (0.51) CA12CA1CA2CA7CA9
SCHEMBL3784304 0.87 ALDH1A1 (0.49) CA12CA1CA2TYRCA7
SCHEMBL3683823 0.87 CA12 (0.51) CA12CA1CA2CA7CA9
SCHEMBL29547544 0.86 NPSR1 (0.46) CA12CA1CA2TYRCA7
SCHEMBL28395325 0.86 CA12 (0.52) CA12CA1CA2CA7CA9
SCHEMBL4619798 0.83 P4HTM (0.53) SMN1; SMN2KDM4EAOC3ALDH1A1NPSR1
SCHEMBL7657058 0.82 P4HTM (0.54) CA12CA1CA2TYRCA7
SCHEMBL7657066 0.82 P4HTM (0.54) CA12CA1CA2TYRCA7
SCHEMBL20128887 0.81 GPR119 (0.52) SMN1; SMN2HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1882687-A1 Heterocyclic compounds useful as vanilloid receptor antagonists and pharmaceutical compositions containing the same Amorepacific Corporation (KR) 2008-01-30 EP disclosed