SCHEMBL4625005

SCHEMBL4625005

COc1ccccc1Oc1ccc2cc(CC(C)(NC(=O)c3c(Cl)cccc3Cl)C(=O)O)ccc2n1

nearest known ligand 0.40

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 4/20 0.40
ITGAV P06756 1/20 0.40
ITGA4 P13612 3/20 0.36
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
NOD2 Q9HC29 1/20 0.35
PKM P14618 1/20 0.35
THRB P10828 1/20 0.35
ITGB7 P26010 1/20 0.34
ALDH1A1 P00352 2/20 0.34
NPSR1 Q6W5P4 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
PTGFR P43088 2/20 0.34
MAPT P10636 2/20 0.34
POLB P06746 1/20 0.33
CASR P41180 1/20 0.33
PTGS2 P35354 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6142440 0.89 ITGB1 (0.42) ITGB1ITGAVITGA4ITGB7ALDH1A1
SCHEMBL4624872 0.86 ITGB1 (0.51) ITGB1ITGAVITGA4ITGB7MAPT
SCHEMBL4624059 0.80 ITGA4 (0.50) ITGB1ITGA4ITGB7ALDH1A1SMN1; SMN2
SCHEMBL4626488 0.80 ITGB1 (0.64) ITGB1ITGAVITGA4ITGB7
SCHEMBL3319930 0.80 ITGB1 (0.61) ITGB1ITGAVITGA4KMT2AITGB7
SCHEMBL4624998 0.78 ITGB1 (0.54) ITGB1ITGAVITGA4ITGB7
SCHEMBL1028112 0.75 ITGB1 (0.55) ITGB1ITGAVITGA4KMT2AITGB7
SCHEMBL4625003 0.73 SMN1; SMN2 (0.41) ITGB1ITGAVITGA4MEN1KMT2A
SCHEMBL4624246 0.73 ITGB1 (0.64) ITGB1ITGAVITGA4ITGB7
SCHEMBL3313216 0.71 ITGB1 (0.50) ITGB1ITGAVITGA4MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501801-B1 2,6-QUINOLINYL AND 2,6-NAPHTHYL DERIVATIVES AND THEIR USE IN THE TREATMENT OF VLA-4 DEPENDENT DISEASES UCB PHARMA SA (BE) 2008-01-23 EP disclosed