SCHEMBL4625235

SCHEMBL4625235

COC(=O)C(Cc1ccc2cc(-c3c(Cl)cccc3Cl)ccc2c1)NC(=O)c1c(Cl)cccc1Cl

nearest known ligand 0.56

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 16/20 0.56
ITGAV P06756 2/20 0.56
ITGA4 P13612 15/20 0.49
ITGB7 P26010 13/20 0.49
HDAC1 Q13547 2/20 0.47
HDAC6 Q9UBN7 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3312750 0.92 ITGA4 (0.58) ITGB1ITGAVITGA4ITGB7HDAC1
SCHEMBL3314241 0.88 ITGB1 (0.70) ITGB1ITGAVITGA4ITGB7
SCHEMBL8353596 0.84 ITGB1 (0.80) ITGB1ITGAVITGA4ITGB7
SCHEMBL3319924 0.84 ITGB1 (0.80) ITGB1ITGAVITGA4ITGB7
SCHEMBL3315770 0.84 ITGB1 (0.80) ITGB1ITGAVITGA4ITGB7
SCHEMBL3314549 0.84 ITGB1 (0.61) ITGB1ITGAVITGA4ITGB7
SCHEMBL3315332 0.81 ALDH1A1 (0.44) ITGB1ITGAVHDAC1HDAC6
SCHEMBL3314284 0.81 TACR1 (0.55) ITGB1ITGAVITGA4ITGB7HDAC1
SCHEMBL20025228 0.81 ITGB1 (0.59) ITGB1ITGAVITGA4ITGB7
SCHEMBL5781376 0.81 ITGA4 (0.70) ITGB1ITGA4ITGB7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20080064720-A1 2,6-Quinolinyl And 2,6-Naphthyl Derivatives, Processes For Preparing Them And Their Uses As Vla-4 Inhibitors UCB, S.A. (BE) 2008-03-13 US disclosed
EP-1501801-B1 2,6-QUINOLINYL AND 2,6-NAPHTHYL DERIVATIVES AND THEIR USE IN THE TREATMENT OF VLA-4 DEPENDENT DISEASES UCB PHARMA SA (BE) 2008-01-23 EP disclosed
EP-1870402-A1 2,6-quinolinyl and 2,6-naphthyl derivatives, processes for preparing them and their uses as VLA-4 inhibitors UCB Pharma, S.A. (BE) 2007-12-26 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080064720-A1 2,6-Quinolinyl And 2,6-Naphthyl Derivatives, Processes For Preparing Them And Their Uses As Vla-4 Inhibitors VCAM1, HRH4, LTA4H ITGB1 781/4885ITGAV 425/4885ITGA4 29/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.