SCHEMBL462576

SCHEMBL462576

CC(C)(C)c1ccc(NC(=S)NN)cc1

nearest known ligand 0.67

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 7/20 0.58
MAPT P10636 6/20 0.58
KDM4E B2RXH2 3/20 0.58
KIF11 P52732 1/20 0.51
HTT P42858 2/20 0.50
LMNA P02545 1/20 0.50
ALOX12 P18054 1/20 0.50
GAA P10253 2/20 0.48
MEN1 O00255 2/20 0.47
KMT2A Q03164 2/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
ALDH1A1 P00352 1/20 0.47
NPC1 O15118 1/20 0.47
XBP1 P17861 1/20 0.47
MAPK1 P28482 1/20 0.47
RAB9A P51151 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31388334 0.88 MAPT (0.55) MAPTKDM4EKIF11HTTLMNA
SCHEMBL455344 0.83 IDO1 (0.78) IDO1MAPTKDM4EGAAMEN1
SCHEMBL457226 0.81 IDO1 (0.65) IDO1MAPTKDM4EKIF11HTT
SCHEMBL28649815 0.81 ALDH1A1 (0.65) MAPTHTTLMNAALOX12GAA
SCHEMBL17465537 0.81 HTT (0.68) MAPTKIF11HTTLMNAALOX12
SCHEMBL4348957 0.80 KIF11 (0.59) MAPTKIF11HTTLMNAALOX12
SCHEMBL23453330 0.78 LMNA (0.58) MAPTKDM4EHTTLMNAALOX12
SCHEMBL455272 0.78 IDO1 (0.64) IDO1MAPTKDM4EHTTGAA
SCHEMBL9037064 0.77 NPC1 (0.66) MAPTKIF11HTTLMNAMEN1
SCHEMBL25494628 0.77 LMNA (0.57) MAPTHTTLMNAALOX12GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013026021-A2 TRKA AS A TARGET FOR INHIBITING APP CLEAVAGE AND/OR PROGRESSION OF ALZHEIMER'S DISEASE BUCK INSTITUTE FOR RESEARCH ON AGING (US) 2013-02-21 WO disclosed
WO-2012033601-A1 THIOSEMICARBAZONES WITH MDR1 - INVERSE ACTIVITY THE UNITED STATES OF AMERICA, AS REPRESENTED BY THE SECRETARY, DEPARTMENT OF HEALTH & HUMAN SERVICES (US) 2012-03-15 WO disclosed