SCHEMBL457226

SCHEMBL457226

NNC(=S)Nc1ccc(C(F)(F)F)cc1

nearest known ligand 0.65

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 6/20 0.65
MAPT P10636 4/20 0.62
KDM4E B2RXH2 2/20 0.62
KIF11 P52732 2/20 0.61
CDK1 P06493 1/20 0.60
ALDH1A1 P00352 2/20 0.57
MEN1 O00255 3/20 0.55
KMT2A Q03164 3/20 0.55
SMN1; SMN2 Q16637 3/20 0.55
LMNA P02545 2/20 0.55
HTT P42858 2/20 0.55
GAA P10253 1/20 0.55
EPHX2 P34913 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9453957 0.88 CDK1 (0.68) MAPTKDM4EKIF11CDK1ALDH1A1
SCHEMBL455344 0.83 IDO1 (0.78) IDO1MAPTKDM4EALDH1A1MEN1
SCHEMBL5438060 0.81 IDO1 (0.70) IDO1MAPTKDM4EALDH1A1MEN1
SCHEMBL18031170 0.81 GAA (0.69) MAPTKDM4EKIF11CDK1ALDH1A1
SCHEMBL462576 0.81 IDO1 (0.58) IDO1MAPTKDM4EKIF11ALDH1A1
SCHEMBL17956747 0.81 KMT2A (0.69) MAPTKDM4EKIF11CDK1ALDH1A1
SCHEMBL12412636 0.81 L3MBTL1 (0.62) MAPTKIF11CDK1ALDH1A1MEN1
SCHEMBL525759 0.80 KIF11 (0.89) KIF11CDK1ALDH1A1MEN1KMT2A
SCHEMBL26156209 0.79 GAA (0.63) MAPTKIF11CDK1ALDH1A1MEN1
SCHEMBL11057676 0.79 KIF11 (0.63) IDO1MAPTKIF11CDK1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 14 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-122010896-A Bicyclol derivative, pharmaceutical composition thereof, preparation method and application thereof 中国医学科学院药物研究所 2026-05-12 CN disclosed
WO-2025046420-A1 COMPOUND TARGETING EGR-1 AND USE THEREOF FOR TREATMENT OF ATOPIC DERMATITIS 주식회사 아제라메디 2025-03-06 WO disclosed
CN-117645560-A Ferulic acid derivative containing amide and preparation method and application thereof 贵州大学 2024-03-05 CN disclosed
CN-114195691-B Ferulic acid derivative containing amide and preparation method and application thereof 贵州大学 2023-10-20 CN disclosed
CN-114195691-A Amide-containing ferulic acid derivative and preparation method and application thereof 贵州大学 2022-03-18 CN disclosed
US-10975048-B2 Composition of 1,3,4-selenadiazole containing compounds with pharmacological activity HANGZHOU JENNIFER BIOTECH CO LTD (CN) 2021-04-13 US disclosed
EP-2240175-B1 COMPOUNDS WITH MDR1-INVERSE ACTIVITY US GOV HEALTH & HUMAN SERV (US) 2013-01-02 EP disclosed
WO-2012033601-A1 THIOSEMICARBAZONES WITH MDR1 - INVERSE ACTIVITY THE UNITED STATES OF AMERICA, AS REPRESENTED BY THE SECRETARY, DEPARTMENT OF HEALTH & HUMAN SERVICES (US) 2012-03-15 WO disclosed
US-20100316655-A1 COMPOUNDS WITH MDR1-INVERSE ACTIVITY INSTITUTE OF ENZYMOLOGY, BIOLOGICAL RESEARCH CENTER, HUNGARIAN ACADEMY OF SCIENCES (HU) 2010-12-16 US disclosed
EP-2240175-A2 COMPOUNDS WITH MDR1-INVERSE ACTIVITY The Government of the United States of America as represented by the Secretary of the Department of Health and Human Services (US) 2010-10-20 EP disclosed
WO-2009102433-A2 COMPOUNDS WITH MDR1-INVERSE ACTIVITY THE GOVERNMENT OF THE UNITED STATES OF AMERICA AS REPRESENTED BY THE SECRETARY OF THE DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 2009-08-20 WO disclosed
US-4871737-A 3-Amino-5-methyl-1H-pyrazole-4-carboxylic acids and esters thereof as anticonvulsants muscle relaxants and anxiolytics A. H. ROBINS COMPANY, INCORPORATED (US) 1989-10-03 US disclosed
EP-0315433-A2 3-amino-5-methyl-1H-pyrazole-4-carboxylic acids and esters thereof as anticonvulsants, muscle relaxants and anxiolytics A.H. ROBINS COMPANY, INCORPORATED (US) 1989-05-10 EP disclosed
US-4826866-A 3-amino-5-methyl-1H-pyrazole-4-carboxylic acids and esters thereof as anticonvulsants, muscle relaxants and anxiolytics A. H. ROBINS COMPANY, INCORPORATED (US) 1989-05-02 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10975048-B2 Composition of 1,3,4-selenadiazole containing compounds with pharmacological activity GPX4, GPX1, SELENOI IDO1 2150/4885MAPT 3810/4885KDM4E 3993/4885
US-20100316655-A1 COMPOUNDS WITH MDR1-INVERSE ACTIVITY ABCC1, ABCB1, ABCC2 IDO1 4305/4885MAPT 4584/4885KDM4E 4412/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.