SCHEMBL4628817

SCHEMBL4628817

CCCOCc1cccc(-c2c(C)cc(C)cc2C)n1.Cc1cc(C)c(-c2cccc(CO)n2)c(C)c1

nearest known ligand 0.35

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HTR7 P34969 2/20 0.33
CRHR1 P34998 2/20 0.32
NOS1 P29475 1/20 0.31
NOS2 P35228 1/20 0.31
GPBAR1 Q8TDU6 1/20 0.31
CYSLTR1 Q9Y271 1/20 0.31
FFAR1 O14842 1/20 0.31
ALDH1A1 P00352 1/20 0.30
LMNA P02545 1/20 0.30
MAPT P10636 1/20 0.30
HPGD P15428 1/20 0.30
MAPK1 P28482 1/20 0.30
HTT P42858 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30
S1PR3 Q99500 1/20 0.30
FFAR4 Q5NUL3 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2071875 0.94 HTR7 (0.36) HTR7CRHR1NOS1NOS2GPBAR1
SCHEMBL2070847 0.85 NOS1 (0.40) HTR7CRHR1NOS1NOS2ALDH1A1
SCHEMBL12640990 0.78 HTR7 (0.40) HTR7NOS1NOS2FFAR1ALDH1A1
SCHEMBL12577773 0.74 HTR7 (0.44) HTR7NOS1NOS2ALDH1A1
SCHEMBL25015240 0.70 NOS1 (0.40) HTR7CRHR1NOS1NOS2ALDH1A1
SCHEMBL2070175 0.70 LTB4R (0.34) HTR7CRHR1NOS1NOS2ALDH1A1
SCHEMBL2070288 0.70 CRHR1 (0.36) HTR7CRHR1NOS1NOS2FFAR1
SCHEMBL2069540 0.69 CRHR1 (0.42) HTR7CRHR1
SCHEMBL3623211 0.69 CCR1 (0.42) HTR7CRHR1NOS1NOS2ALDH1A1
SCHEMBL12577789 0.68 CA12 (0.34) HTR7FFAR1MAPTHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1732541-A4 CYCLIC COMPOUNDS TAKEDA PHARMACEUTICAL (JP) 2008-03-05 EP disclosed
EP-1732541-A2 CYCLIC COMPOUNDS Takeda Pharmaceutical Company Limited (JP) 2006-12-20 EP disclosed
WO-2005099688-A2 CYCLIC COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2005-10-27 WO disclosed