SCHEMBL46312

SCHEMBL46312

Cc1cnc2c(c1)COC(=O)N2C

nearest known ligand 0.35

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
IDH1 O75874 3/20 0.35
MEN1 O00255 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2C9 P11712 1/20 0.33
KMT2A Q03164 1/20 0.33
HTR1A P08908 1/20 0.32
DRD2 P14416 1/20 0.32
HTR2A P28223 1/20 0.32
IDH2 P48735 1/20 0.31
KDM4E B2RXH2 1/20 0.31
ALDH1A1 P00352 1/20 0.31
HPGD P15428 1/20 0.31
HSD17B10 Q99714 1/20 0.31
AVPR1A P37288 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2066345 0.83 HSD17B10 (0.38) IDH1IDH2HSD17B10
SCHEMBL17813511 0.75 IDH1 (0.40) IDH1IDH2KDM4EALDH1A1HPGD
SCHEMBL3516220 0.75 GSK3A (0.33) IDH1
SCHEMBL8629038 0.75 CYP11B2 (0.36) IDH1MEN1KMT2AHTR1ADRD2
SCHEMBL17813510 0.74 PDE3B (0.33)
SCHEMBL46315 0.73 CYP11B2 (0.50) CYP1A2HTR1ADRD2HTR2A
SCHEMBL2067594 0.72 ADRA2A (0.36) CYP1A2CYP2C9HTR1AHTR2A
SCHEMBL31411118 0.72 ADRA2A (0.36) CYP1A2CYP2C9HTR1AHTR2A
SCHEMBL2067239 0.71 IDH1 (0.31) IDH1
SCHEMBL18168056 0.71 IDH1 (0.43) IDH1IDH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011151436-A2 NOVEL COMPOUNDS, METHOD FOR USE THEM AND PHARMACEUTICAL COMPOSITION CONTAINING THEM EUROSCREEN S.A. (BE) 2011-12-08 WO disclosed