SCHEMBL4631479

SCHEMBL4631479

O=C(NCC(=O)Oc1ccccc1)Nc1ccc(-c2ccncc2)cc1

nearest known ligand 0.62

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 8/20 0.62
ROCK1 Q13464 6/20 0.62
HTT P42858 1/20 0.50
CYP19A1 P11511 1/20 0.49
TAAR1 Q96RJ0 1/20 0.48
NAMPT P43490 5/20 0.46
LMNA P02545 1/20 0.46
PPID Q08752 1/20 0.45
POLB P06746 1/20 0.45
STAT3 P40763 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
CASR P41180 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21753692 0.85 EPHX1 (0.52) HTTLMNAPOLBSMN1; SMN2
SCHEMBL15140688 0.79 PORCN (0.64) ROCK2ROCK1HTTLMNAPOLB
SCHEMBL10458464 0.79 POLB (0.50) POLBSMN1; SMN2
SCHEMBL4525925 0.77 ROCK2 (1.00) ROCK2ROCK1HTTNAMPT
SCHEMBL10458465 0.76 KMT2A (0.49) HTTLMNAPOLBSMN1; SMN2
SCHEMBL27744449 0.75 MAPK1 (0.58) ROCK2ROCK1TAAR1NAMPTLMNA
SCHEMBL27723730 0.75 MAPK1 (0.58) ROCK2ROCK1TAAR1NAMPTLMNA
SCHEMBL10458695 0.75 MAPT (0.44) HTTTAAR1NAMPTLMNAPOLB
SCHEMBL10458697 0.75 MAPT (0.44) HTTTAAR1NAMPTLMNAPOLB
SCHEMBL15140925 0.75 ROCK2 (1.00) ROCK2ROCK1HTTNAMPTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1922306-A2 AMIDE DERIVATIVES AS ROCK INHIBITORS Astellas Pharma Inc. (JP) 2008-05-21 EP disclosed
WO-2007026920-A2 AMIDE DERIVATIVES AS ROCK INHIBITORS ASTELLAS PHARMA INC. (JP) 2007-03-08 WO disclosed