SCHEMBL4632635

SCHEMBL4632635

CC1(C)CCCC(Sc2ccccc2C#N)C1

nearest known ligand 0.44

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
DDB1 Q16531 1/20 0.44
CRBN Q96SW2 1/20 0.44
MAOA P21397 3/20 0.36
MAOB P27338 3/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
AR P10275 3/20 0.35
PTPN11 Q06124 1/20 0.32
XDH P47989 1/20 0.32
TSHR P16473 1/20 0.32
MAPT P10636 1/20 0.31
LDHA P00338 2/20 0.31
LDHB P07195 2/20 0.31
TRPA1 O75762 1/20 0.31
BCL2 P10415 1/20 0.30
PGR P06401 1/20 0.30
NR3C2 P08235 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2655839 0.80 MAOA (0.53) DDB1CRBNMAOAMAOBCYP1A2
SCHEMBL4842682 0.77 ALDH1A1 (0.38)
SCHEMBL2538752 0.77 DDB1 (0.53) DDB1CRBNMAOAMAOBCYP1A2
SCHEMBL14595419 0.69 MAOA (0.38) MAOAMAOB
SCHEMBL2579025 0.69 MAOA (0.38) MAOAMAOB
SCHEMBL17784105 0.66 BACE1 (0.32)
SCHEMBL2581431 0.66 MAOB (0.40) MAOAMAOBMAPTTRPA1
SCHEMBL2586878 0.63 MAOA (0.33) DDB1CRBNMAOAMAOBCYP3A4
Acetonitrile SCHEMBL27498741 0.63 TRPA1 (0.59) MAOAMAOBTRPA1
SCHEMBL514630 0.62 CYP1A2 (0.53) DDB1CRBNCYP1A2CYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1924561-A2 6-ARYLALKYLAMINO- 2,3,4,5-TETRAHYDRO-1H-BENZO[D]AZEPINES AS 5-HT2C RECEPTOR AGONISTS Eli Lilly & Company (US) 2008-05-28 EP disclosed
WO-2007028083-A2 6-ARYLALKYLAMINO- 2,3,4,5-TETRAHYDRO-1H-BENZO[D]AZEPINES AS 5-HT2C RECEPTOR AGONISTS ELI LILLY AND COMPANY (US) 2007-03-08 WO disclosed