SCHEMBL4632760

SCHEMBL4632760

CC(=O)Oc1ccccc1C(=O)OCc1cc(C(O)CNC(C)(C)C)ccc1O

nearest known ligand 0.52

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 7/20 0.52
ADRB1 P08588 5/20 0.52
CYP1A2 P05177 1/20 0.52
CYP2D6 P10635 1/20 0.52
TSHR P16473 1/20 0.52
NFKB1 P19838 1/20 0.52
HIF1A Q16665 1/20 0.52
TDP1 Q9NUW8 1/20 0.51
PMP22 Q01453 1/20 0.50
ADRB3 P13945 3/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Albuterol SCHEMBL4632758 0.85 ADRB2 (0.64) ADRB2ADRB1CYP1A2CYP2D6TSHR
SCHEMBL6838978 0.83 ADRB2 (0.66) ADRB2ADRB1CYP1A2CYP2D6TSHR
SCHEMBL12158793 0.83 ADRB2 (0.66) ADRB2ADRB1CYP1A2CYP2D6TSHR
SCHEMBL11289635 0.79 ADRB2 (0.59) ADRB2ADRB1CYP1A2CYP2D6TSHR
SCHEMBL14141543 0.76 ADRB2 (0.62) ADRB2ADRB1CYP1A2CYP2D6TSHR
SCHEMBL11287951 0.76 ADRB2 (0.52) ADRB2ADRB1CYP1A2CYP2D6TSHR
SCHEMBL11286698 0.75 ADRB2 (0.55) ADRB2ADRB1CYP1A2CYP2D6TSHR
SCHEMBL11329853 0.75 PTGS2 (0.54) CYP1A2TSHRTDP1
SCHEMBL4339029 0.74 HTT (0.50) ADRB2ADRB1CYP1A2CYP2D6TSHR
SCHEMBL11277356 0.74 ADRB2 (0.48) ADRB2ADRB1CYP1A2CYP2D6TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1494711-A4 METHODS FOR TREATING CHRONIC OBSTRUCTIVE PULMONARY DISEASE (COPD) ABGENIX INC (US) 2008-05-28 EP disclosed
EP-1494711-A1 METHODS FOR TREATING CHRONIC OBSTRUCTIVE PULMONARY DISEASE (COPD) Abgenix, Inc. (US) 2005-01-12 EP disclosed
WO-2003080117-A1 METHODS FOR TREATING CHRONIC OBSTRUCTIVE PULMONARY DISEASE (COPD) ABGENIX, INC. (US) 2003-10-02 WO disclosed