SCHEMBL4633267

SCHEMBL4633267

CCc1[nH]nc(O)c1Cc1cc(F)c(OC)c(F)c1

nearest known ligand 0.37

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
DBH P09172 1/20 0.34
TTR P02766 1/20 0.33
P2RX7 Q99572 2/20 0.33
SMPD3 Q9NY59 1/20 0.32
HCAR2 Q8TDS4 1/20 0.31
ADORA2A P29274 1/20 0.31
SLC5A1 P13866 1/20 0.31
SLC5A2 P31639 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3783701 0.83 AR (0.37) DBHTTRP2RX7SLC5A1SLC5A2
SCHEMBL4632389 0.80 TAAR1 (0.41) TTRP2RX7SMPD3HCAR2ADORA2A
SCHEMBL4547651 0.68 PTGS2 (0.58) DBH
SCHEMBL12646239 0.67 SLC5A2 (0.36) SLC5A1SLC5A2
SCHEMBL12589092 0.67 SMN1; SMN2 (0.43) DBH
SCHEMBL4633441 0.66 P2RX7 (0.40) TTRP2RX7HCAR2
SCHEMBL3764427 0.63 MAPT (0.50) DBH
SCHEMBL3775407 0.62 MEN1 (0.43)
SCHEMBL3770602 0.62 TAAR1 (0.42) TTRP2RX7SLC5A1SLC5A2
SCHEMBL13548271 0.62 HTR2A (0.44) DBH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1912656-A2 METHODS FOR PREVENTING AND TREATING METABOLIC DISORDERS AND NEW PYRAZOLE-O-GLYCOSIDE DERIVATIVES Boehringer Ingelheim International GmbH (DE) 2008-04-23 EP disclosed
WO-2007014895-A2 METHODS FOR PREVENTING AND TREATING METABOLIC DISORDERS AND NEW PYRAZOLE-O-GLYCOSIDE DERIVATIVES BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2007-02-08 WO disclosed