SCHEMBL4633604

SCHEMBL4633604

O=C(O)Oc1cc2c(NC(=O)c3ccc(CN4CCNCC4)cc3)n[nH]c2s1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 2/20 0.46
IKBKE Q14164 1/20 0.45
TBK1 Q9UHD2 1/20 0.45
KDR P35968 2/20 0.44
F10 P00742 1/20 0.43
KIT P10721 4/20 0.42
FLT3 P36888 2/20 0.42
ABL1 P00519 3/20 0.40
BCR P11274 3/20 0.40
KDM4E B2RXH2 1/20 0.40
ALDH1A1 P00352 1/20 0.40
MAPT P10636 1/20 0.40
RAB9A P51151 1/20 0.40
FGFR1 P11362 1/20 0.40
SLC2A1 P11166 1/20 0.40
HDAC4 P56524 1/20 0.39
KCNH2 Q12809 1/20 0.39
CHRM3 P20309 1/20 0.39
ITGB3 P05106 1/20 0.39
ITGA2B P08514 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4632616 0.93 KDR (0.46) HDAC1TBK1KDRKITFLT3
SCHEMBL4633324 0.93 ABL1 (0.47) HDAC1TBK1KDRF10KIT
SCHEMBL4632623 0.92 ABL1 (0.48) HDAC1TBK1KDRF10KIT
SCHEMBL4631770 0.92 ABL1 (0.48) HDAC1TBK1KDRF10KIT
SCHEMBL4632530 0.88 KDR (0.44) HDAC1KDRKITFLT3ABL1
SCHEMBL4633593 0.87 HDAC1 (0.48) HDAC1IKBKETBK1KDRF10
SCHEMBL4632682 0.82 HDAC6 (0.38) HDAC1KITFLT3FGFR1
SCHEMBL4632607 0.81 HDAC1 (0.49) HDAC1IKBKETBK1KDRFLT3
SCHEMBL4633619 0.81 NPC1 (0.47)
SCHEMBL2431903 0.80 ABL1 (0.58) HDAC1KDRKITFLT3ABL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1711177-B1 1H-THIENO 2,3-c PYRAZOLE DERIVATIVES USEFUL AS KINASE I INHIBITORS PFIZER ITALIA SRL (IT) 2008-05-28 EP claimed