SCHEMBL4634178

SCHEMBL4634178

CCOC(=O)c1cc(N)c2nc(C)n(C)c2c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 2/20 0.43
CA1 P00915 2/20 0.43
CA2 P00918 2/20 0.43
CA7 P43166 2/20 0.43
CA9 Q16790 2/20 0.43
CA14 Q9ULX7 2/20 0.43
LMNA P02545 1/20 0.42
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
MAOA P21397 1/20 0.42
PTGER4 P35408 3/20 0.41
NPC1 O15118 2/20 0.40
ALOX15 P16050 1/20 0.40
RAB9A P51151 1/20 0.40
JMJD6 Q6NYC1 1/20 0.40
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39
GAA P10253 1/20 0.39
HPGD P15428 1/20 0.39
HSD17B10 Q99714 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4664696 0.85 CA12 (0.51) CA12CA1CA2CA7CA9
SCHEMBL4632328 0.80 KMT2A (0.49) LMNAPTGER4NPC1RAB9AKDM4E
SCHEMBL4737793 0.77 KDM4E (0.41) CA12CA1CA2CA7CA9
SCHEMBL5901336 0.75 PPIA (0.47) NPC1ALOX15RAB9AJMJD6ALDH1A1
SCHEMBL14800136 0.75 KDM4E (0.58) LMNACYP1A2NPC1RAB9AKDM4E
SCHEMBL5901208 0.74 CYP3A4 (0.60) LMNACYP1A2CYP3A4NPC1ALOX15
SCHEMBL10895643 0.72 CA12 (0.60) CA12CA1CA2CA7CA9
SCHEMBL23196121 0.72 CA12 (0.45) CA12CA1CA2CA7CA9
SCHEMBL4632945 0.72 TPMT (0.33) NPC1ALOX15KDM4EALDH1A1GAA
SCHEMBL8700664 0.72 LMNA (0.38) CA12CA1CA2CA7CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1926714-A1 ISOTOPICALLY SUBSTITUTED BENZIMIDAZOLE DERIVATIVES Nycomed GmbH (DE) 2008-06-04 EP disclosed
WO-2007023135-A1 ISOTOPICALLY SUBSTITUTED BENZIMIDAZOLE DERIVATIVES NYCOMED GMBH (DE) 2007-03-01 WO disclosed