SCHEMBL4635957

SCHEMBL4635957

O=S(=O)(O)c1c(F)cc(F)cc1Br

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AGTR1 P30556 1/20 0.45
KMT2A Q03164 2/20 0.40
MEN1 O00255 1/20 0.40
MAPT P10636 1/20 0.36
CCR1 P32246 1/20 0.36
CA1 P00915 3/20 0.35
CA2 P00918 3/20 0.35
CA12 O43570 2/20 0.35
CA9 Q16790 2/20 0.35
CA7 P43166 1/20 0.34
CA13 Q8N1Q1 1/20 0.34
ALDH1A1 P00352 3/20 0.33
CES2 O00748 1/20 0.33
CES1 P23141 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
SPR P35270 1/20 0.32
GAA P10253 1/20 0.32
ERN1 O75460 1/20 0.31
PTGES2 Q9H7Z7 1/20 0.31
HTT P42858 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1360908 0.84 CES2 (0.39) AGTR1CA1CA2CA12CA9
Hydrochloric Acid SCHEMBL27308697 0.82 CES2 (0.38) AGTR1CA1CA2CA12CA9
SCHEMBL2775058 0.81 CA1 (0.50) AGTR1KMT2AMEN1MAPTCCR1
SCHEMBL544703 0.79 AGTR1 (0.45) AGTR1KMT2AMEN1MAPTCCR1
SCHEMBL18373564 0.77 CES2 (0.34) AGTR1KMT2AMEN1CA1CA2
SCHEMBL3422434 0.75 ALDH1A1 (0.37) KMT2AMEN1MAPTCA1CA2
SCHEMBL3140914 0.70 CYP3A4 (0.43) CA1CA2CA12CA9CA7
SCHEMBL2775884 0.70 CA1 (0.58) AGTR1CA1CA2CA12CA9
SCHEMBL11871290 0.70 FABP3 (0.35) CA1CA2CA12CA9CA7
Hydrochloric Acid SCHEMBL28280969 0.69 CA12 (0.38) CA1CA2CA12CA7CA13

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1934187-A1 NOVEL BENZIMIDAZOLE AND BENZOTHIAZOLE DERIVATIVES, METHOD FOR PREPARING SAME, USE THEREOF AS DRUGS, PHARMACEUTICAL COMPOSITIONS AND NOVEL USE IN PARTICULAR AS C-MET INHIBITORS Aventis Pharma S.A. (FR) 2008-06-25 EP disclosed
WO-2007036630-A1 NOVEL BENZIMIDAZOLE AND BENZOTHIAZOLE DERIVATIVES, METHOD FOR PREPARING SAME, USE THEREOF AS DRUGS, PHARMACEUTICAL COMPOSITIONS AND NOVEL USE IN PARTICULAR AS C-MET INHIBITORS AVENTIS PHARMA S.A. (FR) 2007-04-05 WO disclosed