SCHEMBL4636262

SCHEMBL4636262

CCOC(=O)c1cnc(-c2ccc(F)cc2)nc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FOS P01100 2/20 0.54
JUN P05412 2/20 0.54
NFKB1 P19838 2/20 0.54
NFKB2 Q00653 2/20 0.54
RELA Q04206 2/20 0.54
MAPT P10636 5/20 0.52
KMT2A Q03164 3/20 0.52
MEN1 O00255 2/20 0.52
CASP3 P42574 1/20 0.52
TRPV1 Q8NER1 1/20 0.52
SENP7 Q9BQF6 1/20 0.52
TRPM8 Q7Z2W7 1/20 0.50
SMN1; SMN2 Q16637 5/20 0.49
ALDH1A1 P00352 9/20 0.49
KDM4E B2RXH2 6/20 0.49
NPC1 O15118 4/20 0.49
RAB9A P51151 4/20 0.49
HPGD P15428 4/20 0.49
MAPK1 P28482 2/20 0.49
GABRA2 P47869 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4949564 0.84 POLB (0.54) FOSJUNNFKB1NFKB2RELA
SCHEMBL8546622 0.84 ALDH1A1 (0.65) FOSJUNNFKB1NFKB2RELA
SCHEMBL27306333 0.84 FOS (0.47) FOSJUNNFKB1NFKB2RELA
SCHEMBL30357866 0.84 MAOB (0.57) FOSJUNNFKB1NFKB2RELA
SCHEMBL2010059 0.84 NPC1 (0.61) FOSJUNNFKB1NFKB2RELA
SCHEMBL29635221 0.83 PDGFRB (0.54) MAPTKMT2AMEN1CASP3SENP7
SCHEMBL5548180 0.83 CDC7 (0.58) FOSJUNNFKB1NFKB2RELA
SCHEMBL9650464 0.82 MAPT (0.46) MAPTKMT2AMEN1SMN1; SMN2ALDH1A1
SCHEMBL7365076 0.82 KMT2A (0.69) MAPTKMT2AMEN1CASP3TRPV1
SCHEMBL5014336 0.81 FOS (0.60) FOSJUNNFKB1NFKB2RELA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1937652-B1 PYRIMIDINE AMIDE COMPOUNDS AS PGDS INHIBITORS AVENTIS PHARMA INC (US) 2014-07-30 EP disclosed
EP-1937652-A1 PYRIMIDINE AMIDE COMPOUNDS AS PGDS INHIBITORS Aventis Pharmaceuticals Inc. (US) 2008-07-02 EP disclosed
WO-2007041634-A1 PYRIMIDINE AMIDE COMPOUNDS AS PGDS INHIBITORS AVENTIS PHARMACEUTICALS INC. (US) 2007-04-12 WO disclosed