SCHEMBL4636702

SCHEMBL4636702

NS(=O)(=O)c1cccc(Cc2ccncc2)c1C(F)(F)F

nearest known ligand 0.41

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CA1 P00915 2/20 0.37
CA2 P00918 2/20 0.37
CA9 Q16790 2/20 0.37
CA12 O43570 1/20 0.37
CA14 Q9ULX7 1/20 0.37
LMNA P02545 1/20 0.36
AR P10275 1/20 0.36
PTGS2 P35354 1/20 0.36
NSD2 O96028 1/20 0.35
MAPK1 P28482 1/20 0.35
PTGES2 Q9H7Z7 2/20 0.35
CYP17A1 P05093 1/20 0.34
CYP11B1 P15538 1/20 0.34
CYP11B2 P19099 1/20 0.34
S1PR1 P21453 1/20 0.34
S1PR3 Q99500 1/20 0.34
NAMPT P43490 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4662891 0.81 CA2 (0.47) CA1CA2CA9CA12CA14
SCHEMBL27702233 0.75 CA2 (0.47) CA1CA2CA9CA12CA14
SCHEMBL20504959 0.72 CA2 (0.42) CA1CA2CA9CA12CA14
SCHEMBL3658845 0.70 CA2 (0.45) CA1CA2CA9CA12LMNA
SCHEMBL14991105 0.69 TTR (0.37) CA1CA2
SCHEMBL2512044 0.69 CA2 (0.46) CA1CA2CA9CA12CA14
SCHEMBL17698980 0.69 PTGES2 (0.45) CA1CA2CA9CA12CA14
SCHEMBL16556192 0.68 CYP19A1 (0.41) LMNACYP17A1CYP11B1CYP11B2NAMPT
SCHEMBL1069769 0.67 PTGES2 (0.42) CA1CA2CA9CA12CA14
SCHEMBL407413 0.67 CA2 (0.50) CA1CA2CA9CA12CA14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1879859-A2 DIARYLSULFONE SULFONAMIDES AND USE THEROF Wyeth a Corporation of the State of Delaware (US) 2008-01-23 EP disclosed
WO-2006124875-A2 DIARYLSULFONE SULFONAMIDES AND USE THEROF WYETH (US) 2006-11-23 WO disclosed