SCHEMBL1069769

SCHEMBL1069769

NS(=O)(=O)c1cccc(-c2ccccc2)c1C(F)(F)F

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGES2 Q9H7Z7 5/20 0.42
CA2 P00918 8/20 0.41
CA1 P00915 7/20 0.41
CA9 Q16790 4/20 0.41
SCN9A Q15858 2/20 0.40
CA4 P22748 2/20 0.40
CA6 P23280 2/20 0.40
CA12 O43570 2/20 0.40
CA5A P35218 2/20 0.40
PTGS1 P23219 1/20 0.40
PTGS2 P35354 1/20 0.40
CYP2C9 P11712 1/20 0.40
CA7 P43166 1/20 0.40
CA14 Q9ULX7 1/20 0.40
CA5B Q9Y2D0 1/20 0.40
F10 P00742 2/20 0.39
PRSS1 P07477 1/20 0.39
PRSS2 P07478 1/20 0.39
PRSS3 P35030 1/20 0.39
STAT3 P40763 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28160333 0.83 PTGS2 (0.47) PTGS1PTGS2STAT3
SCHEMBL28022982 0.83 PTPN1 (0.41) PTGS2
SCHEMBL30211016 0.82 SCN9A (0.51) PTGES2CA2CA1SCN9APTGS1
SCHEMBL4610069 0.82 STAT3 (0.41) PTGES2CA2CA1CA9SCN9A
SCHEMBL27702233 0.82 CA2 (0.47) PTGES2CA2CA1CA9CA4
SCHEMBL7696386 0.81 SCN9A (0.40) PTGES2SCN9ASTAT3
SCHEMBL28022377 0.80 CA2 (0.40) PTGES2CA2CA1CA9SCN9A
SCHEMBL8770171 0.78 SCN9A (0.45) PTGES2CA2CA1SCN9ACA5A
SCHEMBL7696390 0.78 STAT3 (0.39) PTGES2CA2CA1CA9SCN9A
SCHEMBL48885 0.78 CA2 (0.52) CA2CA1CA9SCN9ACA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2451285-A1 PLATELET-ACTIVATING FACTOR RECEPTOR ANTAGONISTS Merck Sharp & Dohme Corp. (US) 2012-05-16 EP claimed
WO-2011005608-A1 PLATELET-ACTIVATING FACTOR RECEPTOR ANTAGONISTS MERCK SHARP & DOHME CORP. (US) 2011-01-13 WO claimed
CN-105102449-B Antiviral compound 豪夫迈·罗氏有限公司 2017-06-13 CN disclosed
EP-2964635-A1 ANTIVIRAL COMPOUNDS F. Hoffmann-La Roche AG (CH) 2016-01-13 EP disclosed
WO-2014135495-A1 ANTIVIRAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2014-09-12 WO disclosed