SCHEMBL4637469

SCHEMBL4637469

N#Cc1ccc(C(F)(F)F)cc1Oc1c[c]ccc1Cl

nearest known ligand 0.44

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
AR P10275 10/20 0.42
SLC6A4 P31645 4/20 0.38
CYP2D6 P10635 2/20 0.38
SLC6A2 P23975 2/20 0.38
NOS2 P35228 2/20 0.38
MRGPRX4 Q96LA9 2/20 0.37
BCAT2 O15382 1/20 0.36
BCAT1 P54687 1/20 0.36
HTR2A P28223 2/20 0.35
KCNH2 Q12809 2/20 0.35
ESRRA P11474 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1692003 0.76 SLC6A4 (0.42) ARSLC6A4HTR2AKCNH2
SCHEMBL2066970 0.72 RXRA (0.47) MRGPRX4
SCHEMBL27583555 0.72 CYP1A2 (0.59)
SCHEMBL952338 0.71 AR (0.65) ARMRGPRX4
SCHEMBL5656320 0.70 AR (0.50) ARSLC6A4CYP2D6SLC6A2NOS2
SCHEMBL25373566 0.69 AR (0.46) ARSLC6A4CYP2D6SLC6A2NOS2
SCHEMBL4672154 0.69 EPAS1 (0.59)
SCHEMBL29837271 0.68 AR (0.47) ARMRGPRX4
SCHEMBL384969 0.68 AR (0.47) ARMRGPRX4
SCHEMBL4638354 0.68 EPAS1 (0.46)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1937632-A1 NOVEL COMPOUNDS Astra Zeneca AB (SE) 2008-07-02 EP claimed
WO-2007039736-A1 NOVEL COMPOUNDS ASTRAZENECA AB (SE) 2007-04-12 WO claimed
EP-1937632-A1 NOVEL COMPOUNDS Astra Zeneca AB (SE) 2008-07-02 EP disclosed
WO-2007039736-A1 NOVEL COMPOUNDS ASTRAZENECA AB (SE) 2007-04-12 WO disclosed