SCHEMBL4638478

SCHEMBL4638478

O=C(C#Cc1nnn(Cc2cc(C(F)(F)F)cc(C(F)(F)F)c2)c1-c1ccccc1)c1ccc(F)cc1

nearest known ligand 0.41

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 2/20 0.41
ALDH1A1 P00352 2/20 0.40
GAA P10253 1/20 0.40
PKM P14618 1/20 0.40
PTGER4 P35408 5/20 0.38
THRB P10828 1/20 0.38
PTGER3 P43115 1/20 0.38
CDC7 O00311 1/20 0.36
TACR1 P25103 2/20 0.36
PTGDR2 Q9Y5Y4 2/20 0.36
CYP19A1 P11511 1/20 0.35
TSHR P16473 1/20 0.35
AKR1C3 P42330 1/20 0.35
AKR1C2 P52895 1/20 0.35
IDO1 P14902 1/20 0.35
TDO2 P48775 1/20 0.35
POLB P06746 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4637822 0.94 ALDH1A1 (0.43) ADORA3ALDH1A1GAAPTGER4PTGER3
SCHEMBL4637770 0.89 ADORA3 (0.46) ADORA3ALDH1A1GAAPTGER4AKR1C3
SCHEMBL4637820 0.87 GAA (0.40) ADORA3ALDH1A1GAAPTGER4TACR1
SCHEMBL4638051 0.84 ALDH1A1 (0.39) ADORA3ALDH1A1GAAPTGER4THRB
SCHEMBL4638558 0.83 ALDH1A1 (0.42) ADORA3ALDH1A1GAAPTGER4PTGER3
SCHEMBL4638482 0.83 ALDH1A1 (0.44) ADORA3ALDH1A1GAAPTGER4CDC7
SCHEMBL4637826 0.79 ALDH1A1 (0.47) ADORA3ALDH1A1GAAPTGER4PTGDR2
SCHEMBL4637811 0.78 GRM2 (0.36) ADORA3ALDH1A1GAAPTGER4THRB
SCHEMBL4637824 0.77 ALDH1A1 (0.44) ADORA3ALDH1A1GAAPTGER4TACR1
SCHEMBL4638520 0.77 ALDH1A1 (0.44) ALDH1A1GAACDC7TACR1CYP19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501808-B1 TACHYKININ RECEPTOR ANTAGONISTS LILLY CO ELI (US) 2008-07-02 EP disclosed