SCHEMBL4637834

SCHEMBL4637834

COc1ccc(OC(F)(F)F)cc1Cn1nnc(C(=O)c2c(-c3ccccc3Cl)noc2COC2CCCCO2)c1-c1cccnc1

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABL1 P00519 2/20 0.33
GPBAR1 Q8TDU6 1/20 0.33
CYP11B1 P15538 2/20 0.33
CYP11B2 P19099 2/20 0.33
HCRTR1 O43613 3/20 0.33
HCRTR2 O43614 3/20 0.33
LMNA P02545 3/20 0.32
MAPK1 P28482 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
TSHR P16473 2/20 0.32
NPSR1 Q6W5P4 1/20 0.32
SCN5A Q14524 1/20 0.31
SCN9A Q15858 1/20 0.31
NPC1 O15118 1/20 0.31
TACR1 P25103 2/20 0.31
MAPT P10636 1/20 0.31
HPGD P15428 1/20 0.31
CFTR P13569 1/20 0.30
PPARG P37231 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4639390 0.89 GLS (0.35) ABL1GPBAR1CYP11B1CYP11B2HCRTR1
SCHEMBL4639447 0.85 IDH1 (0.35) GPBAR1LMNASMN1; SMN2TSHRNPSR1
SCHEMBL4637794 0.84 ALDH1A1 (0.36) HCRTR1HCRTR2LMNAMAPK1SMN1; SMN2
SCHEMBL4637865 0.84 ALDH1A1 (0.33) LMNAMAPK1SMN1; SMN2TSHRNPSR1
SCHEMBL6426240 0.81 ABL1 (0.38) ABL1GPBAR1CYP11B1CYP11B2SMN1; SMN2
SCHEMBL4638945 0.76 IDH1 (0.35) CFTR
SCHEMBL4638641 0.75 IDH1 (0.41) TSHRCFTR
SCHEMBL4637728 0.75 IDH1 (0.37) GPBAR1TSHRTACR1CFTR
SCHEMBL4637757 0.74 ALDH1A1 (0.33) TSHR
SCHEMBL4638099 0.74 IDH1 (0.36) CYP11B1CYP11B2TSHRMAPTCFTR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501808-B1 TACHYKININ RECEPTOR ANTAGONISTS LILLY CO ELI (US) 2008-07-02 EP disclosed