SCHEMBL4637883

SCHEMBL4637883

O=C(C#Cc1nnn(Cc2cc(C(F)(F)F)cc(C(F)(F)F)c2)c1-c1cnccn1)c1ccccc1Cl

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 3/20 0.35
USP2 O75604 4/20 0.35
CYP3A4 P08684 2/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
CYP2D6 P10635 2/20 0.34
IDH1 O75874 1/20 0.34
TACR1 P25103 1/20 0.34
MAPT P10636 2/20 0.33
THRB P10828 1/20 0.33
GRM2 Q14416 1/20 0.33
GPBAR1 Q8TDU6 6/20 0.33
HSD11B1 P28845 1/20 0.33
KDM4E B2RXH2 1/20 0.33
HTT P42858 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
NTRK1 P04629 1/20 0.32
NTRK3 Q16288 1/20 0.32
NTRK2 Q16620 1/20 0.32
TSHR P16473 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4638481 0.88 IDH1 (0.44) P2RX7IDH1TACR1MAPTGRM2
SCHEMBL4637811 0.86 GRM2 (0.36) USP2CYP3A4CYP2D6IDH1TACR1
SCHEMBL4637948 0.86 RORB (0.36) P2RX7IDH1TACR1MAPTTHRB
SCHEMBL4638051 0.85 ALDH1A1 (0.39) TACR1MAPTTHRBGRM2KDM4E
SCHEMBL4637887 0.84 USP2 (0.36) P2RX7USP2CYP3A4MEN1KMT2A
SCHEMBL4637984 0.83 TACR1 (0.39) P2RX7MEN1KMT2ATACR1MAPT
SCHEMBL4638552 0.82 TACR1 (0.40) P2RX7TACR1MAPTTHRBGRM2
SCHEMBL4637750 0.81 IDH1 (0.43) P2RX7CYP3A4MEN1KMT2AIDH1
SCHEMBL4637712 0.81 IDH1 (0.51) P2RX7CYP3A4IDH1MAPTGRM2
SCHEMBL4706074 0.80 RORB (0.39) P2RX7USP2CYP3A4MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501808-B1 TACHYKININ RECEPTOR ANTAGONISTS LILLY CO ELI (US) 2008-07-02 EP disclosed