SCHEMBL4637712

SCHEMBL4637712

O=C(C#Cc1nnn(Cc2ccc(C(F)(F)F)cc2)c1-c1cccnc1)c1ccccc1Cl

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDH1 O75874 1/20 0.51
GRM2 Q14416 1/20 0.38
TEAD1 P28347 1/20 0.38
MAPT P10636 1/20 0.37
SLC2A1 P11166 1/20 0.37
SLC2A3 P11169 1/20 0.37
SLC2A4 P14672 1/20 0.37
HIF1A Q16665 1/20 0.36
EPAS1 Q99814 1/20 0.36
ADORA3 P0DMS8 1/20 0.36
NR3C1 P04150 1/20 0.36
PTGER4 P35408 2/20 0.36
GAA P10253 1/20 0.35
PTGER3 P43115 1/20 0.35
P2RX7 Q99572 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
F2 P00734 1/20 0.35
CYP3A4 P08684 1/20 0.35
S1PR1 P21453 1/20 0.35
PDE4A P27815 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4638481 0.93 IDH1 (0.44) IDH1GRM2MAPTSLC2A1SLC2A3
SCHEMBL4637750 0.92 IDH1 (0.43) IDH1GRM2MAPTADORA3PTGER4
SCHEMBL4638903 0.87 IDH1 (0.38) IDH1GRM2MAPTSLC2A1SLC2A3
SCHEMBL4638808 0.87 P2RX7 (0.38) IDH1MAPTADORA3P2RX7SMN1; SMN2
SCHEMBL4637811 0.85 GRM2 (0.36) IDH1GRM2MAPTHIF1AADORA3
SCHEMBL4637948 0.84 RORB (0.36) IDH1GRM2MAPTADORA3P2RX7
SCHEMBL4638051 0.84 ALDH1A1 (0.39) GRM2MAPTADORA3PTGER4GAA
SCHEMBL4637714 0.83 IDH1 (0.54) IDH1GRM2TEAD1SLC2A1SLC2A3
SCHEMBL4637883 0.81 P2RX7 (0.35) IDH1GRM2MAPTP2RX7SMN1; SMN2
SCHEMBL4637847 0.79 ABL1 (0.40) IDH1MAPTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501808-B1 TACHYKININ RECEPTOR ANTAGONISTS LILLY CO ELI (US) 2008-07-02 EP disclosed