SCHEMBL4638481

SCHEMBL4638481

O=C(C#Cc1nnn(Cc2cc(C(F)(F)F)cc(C(F)(F)F)c2)c1-c1cccnc1)c1ccccc1Cl

nearest known ligand 0.44

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
IDH1 O75874 1/20 0.44
SLC2A1 P11166 1/20 0.36
SLC2A3 P11169 1/20 0.36
SLC2A4 P14672 1/20 0.36
KDR P35968 1/20 0.36
GRM2 Q14416 1/20 0.35
GPBAR1 Q8TDU6 5/20 0.35
GAA P10253 1/20 0.34
P2RX7 Q99572 2/20 0.34
TACR1 P25103 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
F2 P00734 1/20 0.34
MAPT P10636 1/20 0.34
CYP11B1 P15538 1/20 0.34
CYP11B2 P19099 1/20 0.34
S1PR1 P21453 1/20 0.34
CRHR1 P34998 1/20 0.34
RORC P51449 1/20 0.33
RORB Q92753 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4637750 0.94 IDH1 (0.43) IDH1GRM2P2RX7SMN1; SMN2MAPT
SCHEMBL4637712 0.93 IDH1 (0.51) IDH1SLC2A1SLC2A3SLC2A4GRM2
SCHEMBL4637948 0.92 RORB (0.36) IDH1GRM2GPBAR1P2RX7TACR1
SCHEMBL4638051 0.91 ALDH1A1 (0.39) GRM2GAATACR1SMN1; SMN2MAPT
SCHEMBL4637811 0.91 GRM2 (0.36) IDH1GRM2GPBAR1GAATACR1
SCHEMBL4638808 0.89 P2RX7 (0.38) IDH1P2RX7SMN1; SMN2F2MAPT
SCHEMBL4637883 0.88 P2RX7 (0.35) IDH1GRM2GPBAR1P2RX7TACR1
SCHEMBL4638903 0.86 IDH1 (0.38) IDH1SLC2A1SLC2A3SLC2A4KDR
SCHEMBL4638576 0.85 IDH1 (0.41) IDH1KDRGPBAR1GAATACR1
SCHEMBL4637984 0.84 TACR1 (0.39) GRM2GAAP2RX7TACR1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501808-B1 TACHYKININ RECEPTOR ANTAGONISTS LILLY CO ELI (US) 2008-07-02 EP disclosed
EP-1501809-B1 TRIAZOLE DERIVATIVES AS TACHYKININ RECEPTOR ANTAGONISTS LILLY CO ELI (US) 2008-01-16 EP disclosed