SCHEMBL4637945

SCHEMBL4637945

CC(C)(C)[Si](C)(C)OCCc1onc(-c2ccccc2Cl)c1C(=O)c1nnn(Cc2cc(C(F)(F)F)cc(C(F)(F)F)c2)c1Cl

nearest known ligand 0.37

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
EPAS1 Q99814 2/20 0.37
GPBAR1 Q8TDU6 5/20 0.36
MAPT P10636 3/20 0.35
HPGD P15428 2/20 0.35
TSHR P16473 2/20 0.35
ALDH1A1 P00352 2/20 0.34
NLRP3 Q96P20 1/20 0.34
RECQL P46063 1/20 0.34
TACR1 P25103 2/20 0.34
TP53 P04637 1/20 0.33
KMT2A Q03164 2/20 0.33
KDM4E B2RXH2 1/20 0.33
MEN1 O00255 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4637747 0.93 EPAS1 (0.38) EPAS1GPBAR1MAPTHPGDTSHR
SCHEMBL4637843 0.92 GPBAR1 (0.38) EPAS1GPBAR1MAPTHPGDTSHR
SCHEMBL4639007 0.90 GPBAR1 (0.37) EPAS1GPBAR1MAPTHPGDTSHR
SCHEMBL4637922 0.89 TACR1 (0.36) EPAS1GPBAR1MAPTHPGDTSHR
SCHEMBL4638545 0.89 ALDH1A1 (0.38) EPAS1GPBAR1MAPTHPGDTSHR
SCHEMBL4672009 0.88 ALDH1A1 (0.35) EPAS1GPBAR1MAPTHPGDTSHR
SCHEMBL4707134 0.86 EPAS1 (0.40) EPAS1GPBAR1MAPTHPGDTSHR
SCHEMBL4637966 0.84 KMT2A (0.41) MAPTHPGDALDH1A1TACR1TP53
SCHEMBL4637783 0.84 TACR1 (0.41) EPAS1GPBAR1MAPTHPGDTSHR
SCHEMBL4639459 0.83 TACR1 (0.34) EPAS1MAPTTACR1TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501808-B1 TACHYKININ RECEPTOR ANTAGONISTS LILLY CO ELI (US) 2008-07-02 EP disclosed