SCHEMBL4638668

SCHEMBL4638668

O=C(O)c1nnn(Cc2cccc(C(F)(F)F)c2)c1-c1cccnc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 2/20 0.51
GRIN1 Q05586 3/20 0.48
GRIN2B Q13224 3/20 0.48
HTT P42858 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.46
PTGER4 P35408 2/20 0.46
IDH1 O75874 1/20 0.45
TP53 P04637 1/20 0.45
ALDH1A1 P00352 1/20 0.45
GAA P10253 1/20 0.45
MAPT P10636 1/20 0.44
CYP11B1 P15538 1/20 0.44
CYP11B2 P19099 1/20 0.44
SORT1 Q99523 1/20 0.44
CYP19A1 P11511 1/20 0.43
AKR1C3 P42330 1/20 0.43
AKR1C2 P52895 1/20 0.43
P2RX7 Q99572 1/20 0.43
P2RY14 Q15391 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4637742 0.92 ALDH1A1 (0.52) POLBGRIN1GRIN2BIDH1ALDH1A1
SCHEMBL27606659 0.90 POLB (0.49) POLBGRIN1GRIN2BHTTL3MBTL1
SCHEMBL4638551 0.89 IDH1 (0.55) POLBPTGER4IDH1ALDH1A1GAA
SCHEMBL4637730 0.88 MAPT (0.50) POLBGRIN1GRIN2BHTTL3MBTL1
SCHEMBL4639523 0.85 MAPT (0.46) POLBGRIN1GRIN2BHTTL3MBTL1
SCHEMBL4637958 0.85 POLB (0.45) POLBGRIN1GRIN2BIDH1ALDH1A1
SCHEMBL4637702 0.82 PTGER4 (0.44) GRIN1GRIN2BL3MBTL1PTGER4IDH1
N-Benzylmethylamine SCHEMBL5796449 0.82 POLB (0.54) POLBHTTL3MBTL1SMN1; SMN2PTGER4
SCHEMBL4637753 0.82 IDH1 (0.47) POLBGRIN1GRIN2BHTTL3MBTL1
SCHEMBL27625194 0.81 IDH1 (0.51) POLBPTGER4IDH1ALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501808-B1 TACHYKININ RECEPTOR ANTAGONISTS LILLY CO ELI (US) 2008-07-02 EP disclosed