SCHEMBL4638835

SCHEMBL4638835

Clc1ccccc1-c1coc(C2CC2)n1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 1/20 0.38
HSP90AB1 P08238 1/20 0.38
ALDH1A1 P00352 3/20 0.38
HTT P42858 2/20 0.38
TSHR P16473 1/20 0.38
CYP19A1 P11511 1/20 0.38
IDO1 P14902 1/20 0.38
CHRNB2 P17787 1/20 0.38
CHRNA4 P43681 1/20 0.38
SMN1; SMN2 Q16637 2/20 0.37
LMNA P02545 1/20 0.37
MAPT P10636 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
HCRTR2 O43614 1/20 0.37
ABL1 P00519 3/20 0.37
NPC1 O15118 1/20 0.37
TP53 P04637 1/20 0.37
HPGD P15428 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19399205 0.76 HCRTR2 (0.48) ALDH1A1MAPTL3MBTL1HCRTR2NPC1
SCHEMBL4638064 0.73 ENPP3 (0.55) HSP90AA1HSP90AB1ALDH1A1CYP19A1IDO1
SCHEMBL30263376 0.73 HSP90AA1 (0.50) HSP90AA1HSP90AB1ALDH1A1CYP19A1IDO1
SCHEMBL24107475 0.73 HSP90AA1 (0.50) HSP90AA1HSP90AB1ALDH1A1CYP19A1IDO1
SCHEMBL30605718 0.69 STAT3 (0.52) ALDH1A1HTTCHRNB2CHRNA4SMN1; SMN2
SCHEMBL4639385 0.69 HSP90AA1 (0.39) HSP90AA1HSP90AB1CYP19A1IDO1SMN1; SMN2
SCHEMBL4638829 0.69 NPC1 (0.40) ALDH1A1HTTTSHRSMN1; SMN2LMNA
SCHEMBL20501614 0.68 IDO1 (0.41) CYP19A1IDO1HCRTR2CLK4
Hydrochloric Acid SCHEMBL30605737 0.68 STAT3 (0.51) ALDH1A1HTTCHRNB2CHRNA4SMN1; SMN2
SCHEMBL21834023 0.66 ALDH1A1 (0.44) ALDH1A1TSHRLMNAMAPTHCRTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501808-B1 TACHYKININ RECEPTOR ANTAGONISTS LILLY CO ELI (US) 2008-07-02 EP disclosed
CN-1649849-A Tachykinin receptor antagonists LILLY CO ELI (US) 2005-08-03 CN disclosed