SCHEMBL4640487

SCHEMBL4640487

COC(=O)Oc1ccc2c(c1)[nH]c(=O)n2CCC(C)(C)N

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.41
MEN1 O00255 2/20 0.41
RAB9A P51151 1/20 0.41
CALCRL Q16602 1/20 0.39
HPGD P15428 4/20 0.37
EPHX2 P34913 3/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
PPARG P37231 2/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
MAOB P27338 1/20 0.36
KDM4E B2RXH2 4/20 0.35
ALDH1A1 P00352 3/20 0.35
GLA P06280 3/20 0.35
GAA P10253 3/20 0.35
HSD17B10 Q99714 3/20 0.35
PKM P14618 1/20 0.34
HTT P42858 1/20 0.34
POLB P06746 2/20 0.34
TSHR P16473 1/20 0.34
MDM2 Q00987 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4640794 0.89 MEN1 (0.38) KMT2AMEN1RAB9ACALCRLHPGD
SCHEMBL4640997 0.83 MEN1 (0.36) KMT2AMEN1RAB9ACALCRLHPGD
SCHEMBL4915808 0.82 KDM4E (0.53) KMT2AMEN1RAB9AHPGDSMN1; SMN2
SCHEMBL1858719 0.74 MAPT (0.47) KMT2AMEN1MAOBKDM4EALDH1A1
SCHEMBL13082395 0.74 MEN1 (0.35) KMT2AMEN1RAB9AHPGDSMN1; SMN2
SCHEMBL4604850 0.74 MTNR1A (0.50) KMT2AMEN1RAB9ASMN1; SMN2MAOB
SCHEMBL739035 0.73 MEN1 (0.59) KMT2AMEN1RAB9AHPGDSMN1; SMN2
SCHEMBL8125879 0.70 KMO (0.55) KMT2AMEN1CALCRLHPGDEPHX2
Trifluoroacetic Acid SCHEMBL4607803 0.70 MEN1 (0.49) KMT2AMEN1RAB9AHPGDSMN1; SMN2
SCHEMBL1858977 0.70 DAO (0.50) KMT2AMEN1CALCRLHPGDSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1943229-A1 BENZIMIDAZOLE DERIVATIVES FOR USE AS BETA-3 RECEPTOR AGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2008-07-16 EP disclosed
WO-2007048842-A1 BENZIMIDAZOLE DERIVATIVES FOR USE AS BETA-3 RECEPTOR AGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2007-05-03 WO disclosed