SCHEMBL4640568

SCHEMBL4640568

CCOc1cccnc1CC(=O)Cc1coc(-c2ccc(OC)c(OC3CCCC3)c2)n1

nearest known ligand 0.47

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 17/20 0.43
PDE4B Q07343 13/20 0.43
PDE4C Q08493 13/20 0.43
PDE4D Q08499 13/20 0.43
S1PR1 P21453 1/20 0.43
S1PR3 Q99500 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4639397 0.90 PDE4A (0.44) PDE4APDE4BPDE4CPDE4DS1PR1
SCHEMBL4639574 0.85 MAPT (0.37) S1PR1S1PR3
SCHEMBL4281121 0.83 S1PR1 (0.43) PDE4APDE4BPDE4CPDE4DS1PR1
SCHEMBL4284194 0.83 PDE4A (0.45) PDE4APDE4BPDE4CPDE4DS1PR1
SCHEMBL4639603 0.82 PDE4A (0.44) PDE4APDE4BPDE4CPDE4DS1PR1
SCHEMBL4279424 0.80 PDE4A (0.44) PDE4APDE4BPDE4CPDE4DS1PR1
SCHEMBL4641099 0.80 PDE4A (0.39) PDE4APDE4BPDE4CPDE4D
SCHEMBL4277016 0.79 S1PR1 (0.45) PDE4APDE4BPDE4CPDE4DS1PR1
SCHEMBL4284494 0.79 PDE4A (0.46) PDE4APDE4BPDE4CPDE4D
SCHEMBL4639813 0.78 S1PR1 (0.43) S1PR1S1PR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1954684-A2 OXAZOLE COMPOUND AND PHARMACEUTICAL COMPOSITION Otsuka Pharmaceutical Co., Ltd. (JP) 2008-08-13 EP disclosed
WO-2007058338-A9 OXAZOLE COMPOUND AND PHARMACEUTICAL COMPOSITION OTSUKA PHARMA CO LTD (JP) 2007-11-01 WO disclosed
WO-2007058338-A2 OXAZOLE COMPOUND AND PHARMACEUTICAL COMPOSITION OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2007-05-24 WO disclosed