SCHEMBL4642278

SCHEMBL4642278

CCOC(=O)Oc1cc2ncn(CCC(C)(C)NC(=O)OC(C)(C)C)c2cc1Cl

nearest known ligand 0.39

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.39
POLB P06746 1/20 0.39
MAPT P10636 1/20 0.39
CDK9 P50750 2/20 0.38
CUL4A Q13619 1/20 0.35
AAK1 Q2M2I8 8/20 0.35
PRPS1 P60891 1/20 0.34
TNF P01375 3/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
BRD4 O60885 1/20 0.33
MTNR1A P48039 1/20 0.32
MTNR1B P49286 1/20 0.32
HSD17B13 Q7Z5P4 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4914665 0.86 ALDH1A1 (0.40) ALDH1A1POLBMAPTCDK9AAK1
SCHEMBL4640617 0.84 ALDH1A1 (0.40) ALDH1A1POLBMAPTCDK9AAK1
SCHEMBL4641222 0.84 MTNR1A (0.45) ALDH1A1POLBMAPTCDK9AAK1
SCHEMBL4768461 0.84 ALDH1A1 (0.38) ALDH1A1POLBMAPTCDK9AAK1
SCHEMBL4641876 0.82 AAK1 (0.35) ALDH1A1CDK9AAK1PRPS1TNF
SCHEMBL4648898 0.81 BRD4 (0.35) ALDH1A1CDK9AAK1PRPS1BRD4
SCHEMBL4640258 0.79 BRD4 (0.35) ALDH1A1POLBMAPTCDK9AAK1
SCHEMBL4890412 0.78 ALDH1A1 (0.39) ALDH1A1POLBMAPTCDK9TNF
SCHEMBL4911401 0.78 NPC1 (0.45) ALDH1A1POLBMAPTCDK9NPC1
SCHEMBL4887298 0.78 ALDH1A1 (0.39) ALDH1A1POLBMAPTCDK9TNF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1943229-A1 BENZIMIDAZOLE DERIVATIVES FOR USE AS BETA-3 RECEPTOR AGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2008-07-16 EP disclosed
WO-2007048842-A1 BENZIMIDAZOLE DERIVATIVES FOR USE AS BETA-3 RECEPTOR AGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2007-05-03 WO disclosed