SCHEMBL4768461

SCHEMBL4768461

CCOC(=O)Oc1cc2ncn(CCC(C)(C)NC(=O)OC(C)(C)C)c2cn1

nearest known ligand 0.38

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.38
MAPT P10636 3/20 0.38
POLB P06746 2/20 0.38
CDK9 P50750 1/20 0.33
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32
TNF P01375 4/20 0.32
HDAC1 Q13547 1/20 0.32
BRD4 O60885 1/20 0.31
TP53 P04637 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
MTNR1A P48039 1/20 0.31
MTNR1B P49286 1/20 0.31
HPGD P15428 1/20 0.31
AAK1 Q2M2I8 2/20 0.30
LMNA P02545 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4887298 0.85 ALDH1A1 (0.39) ALDH1A1MAPTPOLBCDK9NPC1
SCHEMBL4642278 0.84 ALDH1A1 (0.39) ALDH1A1MAPTPOLBCDK9NPC1
SCHEMBL4775013 0.83 ALDH1A1 (0.38) ALDH1A1MAPTPOLBCDK9NPC1
SCHEMBL4641222 0.83 MTNR1A (0.45) ALDH1A1MAPTPOLBCDK9NPC1
SCHEMBL4890412 0.79 ALDH1A1 (0.39) ALDH1A1MAPTPOLBCDK9NPC1
SCHEMBL4907499 0.79 NPC1 (0.45) ALDH1A1MAPTPOLBNPC1RAB9A
SCHEMBL4640258 0.78 BRD4 (0.35) ALDH1A1MAPTPOLBCDK9TNF
SCHEMBL4914665 0.77 ALDH1A1 (0.40) ALDH1A1MAPTPOLBCDK9NPC1
SCHEMBL4641876 0.77 AAK1 (0.35) ALDH1A1CDK9TNFBRD4HPGD
SCHEMBL4640617 0.77 ALDH1A1 (0.40) ALDH1A1MAPTPOLBCDK9NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1945304-A2 IMIDAZO-PYRIDINE CONTAINING BETA AGONISTS, METHOD FOR PRODUCING THEM AND THEIR USE AS DRUGS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2008-07-23 EP disclosed
WO-2007048843-A2 IMIDAZO-PYRIDINE CONTAINING BETA AGONISTS, METHOD FOR PRODUCING THEM AND THEIR USE AS DRUGS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2007-05-03 WO disclosed