SCHEMBL4642439

SCHEMBL4642439

Clc1ccc2c(c1)CCC=C2c1ncc[nH]1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B2 P19099 11/20 0.39
CYP11B1 P15538 8/20 0.39
CYP19A1 P11511 7/20 0.39
HTT P42858 1/20 0.38
CYP3A4 P08684 4/20 0.38
MEN1 O00255 1/20 0.36
LMNA P02545 1/20 0.36
ADRB2 P07550 1/20 0.36
CHRM2 P08172 1/20 0.36
CHRM4 P08173 1/20 0.36
ABCB1 P08183 1/20 0.36
HTR1A P08908 1/20 0.36
CHRM5 P08912 1/20 0.36
ADRA2A P08913 1/20 0.36
CHRM1 P11229 1/20 0.36
DRD2 P14416 1/20 0.36
ADRA2B P18089 1/20 0.36
ADRA2C P18825 1/20 0.36
CHRM3 P20309 1/20 0.36
DRD1 P21728 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4640789 0.83 ADRA2A (0.41) CYP11B2CYP11B1CYP19A1CYP3A4ADRA2A
SCHEMBL779679 0.80 NISCH (0.43) CYP11B2CYP11B1CYP19A1MEN1ADRA2A
SCHEMBL3631532 0.72 RAB9A (0.50) MEN1KMT2ANPC1RAB9A
SCHEMBL767558 0.71 ADRA2A (0.57) CYP19A1HTTCYP3A4MEN1LMNA
SCHEMBL2776743 0.71 SMPD3 (0.41) ABCB1ADRA2AADRA2CMC4RADRA1A
SCHEMBL31429694 0.71 IDO1 (0.51) CYP19A1CYP3A4NPC1RAB9A
SCHEMBL8542466 0.71 ALDH1A1 (0.49) CYP19A1CYP3A4HTR2BNPC1RAB9A
SCHEMBL9265577 0.70 CYP11B2 (0.39) CYP11B2CYP11B1CYP19A1HTTCYP3A4
SCHEMBL14969027 0.69 NISCH (0.37) ADRA2AADRA1A
SCHEMBL8537063 0.69 NR4A2 (0.43) CYP3A4NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1804805-A4 USE OF AROMATASE INHIBITORS FOR THE TREATMENT OF ECTOPIC PREGNANCY UNIV WAYNE STATE (US) 2008-08-13 EP disclosed
EP-1804805-A2 USE OF AROMATASE INHIBITORS FOR THE TREATMENT OF ECTOPIC PREGNANCY WAYNE STATE UNIVERSITY (US) 2007-07-11 EP disclosed
WO-2006041941-A2 USE OF AROMATASE INHIBITORS FOR THE TREATMENT OF ECTOPIC PREGNANCY WAYNE STATE UNIVERSITY (US) 2006-04-20 WO disclosed