SCHEMBL4643855

SCHEMBL4643855

CN(C)CCN(C)c1nc2cc(NC(=O)Oc3ccc(-c4ccc(Cl)cc4Cl)cc3)ccc2o1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AGPAT2 O15120 6/20 0.45
MAPT P10636 6/20 0.43
KDR P35968 2/20 0.43
CASP3 P42574 1/20 0.42
SENP8 Q96LD8 1/20 0.42
SENP7 Q9BQF6 1/20 0.42
SENP6 Q9GZR1 1/20 0.42
PARP3 Q9Y6F1 1/20 0.42
RXFP1 Q9HBX9 1/20 0.42
THRB P10828 1/20 0.42
MCHR1 Q99705 3/20 0.41
MCHR2 Q969V1 1/20 0.41
CETP P11597 2/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
KDM4E B2RXH2 1/20 0.41
USP2 O75604 1/20 0.41
ALDH1A1 P00352 1/20 0.41
HPGD P15428 1/20 0.41
TSHR P16473 1/20 0.41
MAPK1 P28482 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4641336 0.94 AGPAT2 (0.46) AGPAT2MAPTKDRCASP3SENP8
SCHEMBL4641167 0.92 AGPAT2 (0.46) AGPAT2MAPTTHRB
SCHEMBL13054281 0.87 MAPT (0.54) MAPTKDRRXFP1THRBMCHR1
Hydrochloric Acid SCHEMBL5249492 0.86 MAPT (0.53) MAPTKDRRXFP1THRBMCHR1
SCHEMBL4643568 0.86 MCHR1 (0.47) AGPAT2MAPTKDRRXFP1MCHR1
SCHEMBL4641580 0.85 MAPT (0.48) MAPTRXFP1THRBMCHR1CETP
SCHEMBL4643045 0.83 CHRM3 (0.40) AGPAT2MAPTKDRCASP3SENP8
SCHEMBL5244630 0.81 MAPT (0.53) MAPTKDRRXFP1THRBMCHR1
SCHEMBL4641201 0.81 AGPAT2 (0.42) AGPAT2MAPTKDRCASP3SENP8
SCHEMBL4643578 0.81 MCHR1 (0.44) MAPTMCHR1MCHR2SMN1; SMN2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1828177-B1 NOVEL MCH RECEPTOR ANTAGONISTS LILLY CO ELI (US) 2008-08-13 EP claimed