SCHEMBL4641201

SCHEMBL4641201

CN1CCC(N(C)c2nc3cc(NC(=O)Oc4ccc(-c5ccc(Cl)cc5Cl)cc4)ccc3o2)CC1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AGPAT2 O15120 5/20 0.42
MAPT P10636 6/20 0.40
ROCK2 O75116 1/20 0.39
THRB P10828 1/20 0.39
KDR P35968 1/20 0.38
KDM4E B2RXH2 1/20 0.38
USP2 O75604 1/20 0.38
ALDH1A1 P00352 1/20 0.38
HPGD P15428 1/20 0.38
TSHR P16473 1/20 0.38
MAPK1 P28482 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
HSD17B10 Q99714 1/20 0.38
PTGDR2 Q9Y5Y4 3/20 0.37
POLB P06746 2/20 0.37
CASP3 P42574 2/20 0.37
SENP7 Q9BQF6 2/20 0.37
SLC2A1 P11166 1/20 0.37
SENP8 Q96LD8 1/20 0.37
SENP6 Q9GZR1 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4641410 0.95 AGPAT2 (0.42) AGPAT2MAPTROCK2THRBKDR
SCHEMBL4643048 0.93 AGPAT2 (0.42) AGPAT2MAPTTHRBPOLB
SCHEMBL4643098 0.92 MAPT (0.46) AGPAT2MAPTKDM4EALDH1A1HPGD
SCHEMBL13054298 0.88 MAPT (0.49) MAPTTHRBKDRPOLBSLC2A1
Hydrochloric Acid SCHEMBL5249326 0.88 MAPT (0.49) MAPTTHRBKDRPOLBSLC2A1
SCHEMBL4641300 0.87 AGPAT2 (0.42) AGPAT2MAPTTHRBKDRKDM4E
SCHEMBL4641368 0.87 PTGDR2 (0.40) MAPTTHRBPTGDR2POLB
SCHEMBL4643045 0.87 CHRM3 (0.40) AGPAT2MAPTTHRBKDRKDM4E
SCHEMBL4646624 0.86 MAPT (0.42) MAPTTHRBKDM4EALDH1A1HPGD
SCHEMBL4644568 0.83 CASP3 (0.39) AGPAT2MAPTTHRBKDRPTGDR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1828177-B1 NOVEL MCH RECEPTOR ANTAGONISTS LILLY CO ELI (US) 2008-08-13 EP claimed