SCHEMBL464496

SCHEMBL464496

Fc1ccc(-c2c[nH]cn2)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 2/20 0.40
SMN1; SMN2 Q16637 2/20 0.39
POLB P06746 1/20 0.39
KDM5B Q9UGL1 1/20 0.39
RAB9A P51151 5/20 0.39
NPC1 O15118 5/20 0.39
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
ALDH1A1 P00352 3/20 0.38
ALOX5 P09917 1/20 0.38
ATM Q13315 2/20 0.38
RXFP1 Q9HBX9 1/20 0.38
MAPK13 O15264 1/20 0.37
RAF1 P04049 1/20 0.37
MAPK9 P45984 1/20 0.37
MAPK12 P53778 1/20 0.37
MAPK11 Q15759 1/20 0.37
MAPK14 Q16539 1/20 0.37
SCN4A P35499 1/20 0.37
CA12 O43570 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1384144 0.89 SCN4A (0.53) MEN1KMT2AALDH1A1SCN4AMAPT
SCHEMBL20054187 0.86 AKT1 (0.30)
SCHEMBL25081050 0.82 MAOB (0.51) RAB9ANPC1CA12MAOBCASP3
Butylamine SCHEMBL8653267 0.82 TLR8 (0.44) MEN1KMT2AALDH1A1MAPK13MAPK12
SCHEMBL856079 0.78 METAP2 (0.44) MAPK1SMN1; SMN2RAB9ANPC1MEN1
SCHEMBL5478060 0.78 METAP2 (0.44) MAPK1SMN1; SMN2POLBRAB9ANPC1
SCHEMBL4379353 0.78 IDO1 (0.39)
SCHEMBL1501981 0.78 MAPT (0.45) MAPK1SMN1; SMN2POLBRAB9ANPC1
SCHEMBL13514507 0.78 METAP2 (0.44)
SCHEMBL4063789 0.78 AKT1 (0.43) SMN1; SMN2POLBRAB9ANPC1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 143 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2025132825-A1 1H-IMIDAZO[4,5-C]QUINOLINE METAL-BASED COMPLEXES USEFUL AS MEDICAMENTS FUNDACIÓN DONOSTIA INTERNATIONAL PHYSICS CENTER - DIPC (ES) 2025-06-26 WO claimed
EP-3500562-B1 SUBSTITUTED AZOLE DERIVATIVES FOR GENERATION, PROLIFERATION AND DIFFERENTIATION OF HEMATOPOIETIC STEM AND PROGENITOR CELLS NAT UNIV SINGAPORE (SG) 2023-11-15 EP claimed
US-20140031289-A1 POLY(ORGANOPHOSPHAZENE) CONTAINING DEGRADATION CONTROLLABLE IONIC GROUP, PREPARATION METHOD THEREOF AND USE THEREOF KOREA INSTITUTE OF SCIENCE AND TECHNOLOGY (KR) 2014-01-30 US claimed
US-20110136796-A1 IDO Inhibitors NEWLINK GENETICS (US) 2011-06-09 US claimed
EP-4323354-B1 2-((4-((S)-2-(4-CHLORO-2-FLUOROPHENYL)-2-METHYLBENZO[D][1,3]DIOXOL-4-YL)PIPERIDIN-1-YL)METHYL)-1-(((S)-OXETAN-2-YL)METHYL)-1H-IMIDAZOLE DERIVATIVES AS ACTIVATORS OF THE GLP1 RECEPTOR FOR THE TREATMENT OF OBESITY NOVARTIS AG (CH) 2025-12-17 EP disclosed
WO-2025236011-A1 COMPOSITIONS FOR PHOSPHOROUS-AZOLE EXCHANGE CHEMISTRY AND USE THEREOF TO TARGET FUNCTIONAL PROTEIN SITES BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM (US) 2025-11-13 WO disclosed
EP-4577524-A1 METHODS OF MANUFACTURING KINASE INHIBITORS Insilico Medicine IP Limited (HK) 2025-07-02 EP disclosed
WO-2025132825-A1 1H-IMIDAZO[4,5-C]QUINOLINE METAL-BASED COMPLEXES USEFUL AS MEDICAMENTS FUNDACIÓN DONOSTIA INTERNATIONAL PHYSICS CENTER - DIPC (ES) 2025-06-26 WO disclosed
US-20250197583-A1 THERMALLY TREATED POLYAMIC AMIDE AEROGEL Blueshift Materials, Inc. (US) 2025-06-19 US disclosed
US-20250179059-A1 ANTICANCER COMPOUNDS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA 2025-06-05 US disclosed
CN-119923387-A Method for producing kinase inhibitors 英矽智能科技知识产权有限公司 2025-05-02 CN disclosed
US-20250109270-A1 THERMALLY TREATED POLYAMIC AMIDE AEROGEL Blueshift Materials, Inc. 2025-04-03 US disclosed
US-6100404-A Erythromycin compounds HOECHST MARION ROUSSEL (FR) 2000-08-08 US disclosed
CN-1052984-C Novel erythromycin derivatives, process for their preparation and their use as medicaments ROUSSEL UCLAF (FR) 2000-05-31 CN disclosed
CN-1229082-A Amine compound and its acid addition salt ROUSSEL UCLAF (FR) 1999-09-22 CN disclosed
EP-0680967-B1 Erythromycin derivatives, their process of preparation and their use as medicaments HOECHST MARION ROUSSEL INC (FR) 1998-10-14 EP disclosed
CN-1151746-A Novel erythromycin derivatives, process for their preparation and their use as medicaments ROUSSEL UCLAF (FR) 1997-06-11 CN disclosed
US-5635485-A Erythromycin compounds ROUSSEL UCLAF (FR) 1997-06-03 US disclosed
WO-1995029929-A1 NOVEL ERYTHROMYCIN DERIVATIVES, METHOD FOR THEIR PREPARATION AND THEIR USE AS DRUGS ROUSSEL UCLAF (FR) 1995-11-09 WO disclosed
EP-0680967-A1 Erythromycin derivatives, their process of preparation and their use as medicaments ROUSSEL-UCLAF (FR) 1995-11-08 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250179059-A1 ANTICANCER COMPOUNDS BET1, BRD4, BICRA MAPK1 2457/4885SMN1; SMN2 4326/4885POLB 594/4885
US-20140031289-A1 POLY(ORGANOPHOSPHAZENE) CONTAINING DEGRADATION CONTROLLABLE IONIC GROUP, PREPARATION METHOD THEREOF AND USE THEREOF PHOSPHO1, PLCB3, INPP5D MAPK1 1786/4885SMN1; SMN2 2329/4885POLB 889/4885
US-20110136796-A1 IDO Inhibitors IDO1, IDO2, INMT MAPK1 2450/4885SMN1; SMN2 4704/4885POLB 2996/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.