SCHEMBL4646402

SCHEMBL4646402

O=C(NC(c1ncccc1O)C1CCC1)c1ccc(Cl)cc1Cl

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A9 P48067 6/20 0.47
RAB9A P51151 5/20 0.44
NPC1 O15118 4/20 0.44
ALDH1A1 P00352 3/20 0.42
HPGD P15428 1/20 0.42
JAK2 O60674 1/20 0.42
JAK1 P23458 1/20 0.42
TYK2 P29597 1/20 0.42
TRPM8 Q7Z2W7 1/20 0.41
KMT2A Q03164 3/20 0.41
NSD2 O96028 2/20 0.40
SETD2 Q9BYW2 2/20 0.40
MEN1 O00255 2/20 0.40
GAA P10253 2/20 0.40
ALOX12 P18054 1/20 0.39
NCOA1 Q15788 1/20 0.39
NCOA3 Q9Y6Q9 1/20 0.39
CES1 P23141 1/20 0.39
MAPT P10636 1/20 0.39
MAPK1 P28482 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4645715 0.88 SLC6A9 (0.47) SLC6A9RAB9ANPC1ALDH1A1HPGD
SCHEMBL3059626 0.71 SLC6A9 (0.60) SLC6A9RAB9ANPC1ALDH1A1HPGD
SCHEMBL3055700 0.70 SLC6A9 (0.59) SLC6A9RAB9ANPC1ALDH1A1HPGD
SCHEMBL3059786 0.68 SLC6A9 (0.63) SLC6A9HPGDKMT2AMEN1
SCHEMBL2850005 0.67 SLC6A9 (0.54) SLC6A9RAB9ANPC1ALDH1A1KMT2A
SCHEMBL13754447 0.66 ALDH1A1 (0.72) RAB9ANPC1ALDH1A1HPGDJAK2
SCHEMBL4643557 0.66 KDM4E (0.47) RAB9ANPC1ALDH1A1HPGDJAK2
SCHEMBL2458645 0.66 SLC6A12 (0.46) RAB9ANPC1ALDH1A1HPGDKMT2A
SCHEMBL2460613 0.65 RAB9A (0.47) RAB9ANPC1ALDH1A1HPGDJAK2
SCHEMBL29077678 0.65 HPGD (0.71) RAB9ANPC1ALDH1A1HPGDMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1960360-A1 AZETIDINE DERIVATIVES AS GLYT1 INHIBITORS MERCK SHARP & DOHME LTD. (GB) 2008-08-27 EP disclosed
WO-2007060484-A1 AZETIDINE DERIVATIVES AS GLYT1 INHIBITORS MERCK SHARP & DOHME LIMITED (GB) 2007-05-31 WO disclosed