Timoprazole

Timoprazole

SCHEMBL464728

[O-][S+](Cc1ccccn1)c1nc2ccccc2[nH]1

nearest known ligand 0.51

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 3/20 0.51
CYP2E1 P05181 3/20 0.51
CYP2C8 P10632 3/20 0.51
CYP2D6 P10635 3/20 0.51
CYP2C9 P11712 3/20 0.51
CYP2B6 P20813 3/20 0.51
CYP2C19 P33261 3/20 0.51
RAB9A P51151 6/20 0.44
NPC1 O15118 5/20 0.44
SMN1; SMN2 Q16637 3/20 0.44
PKM P14618 3/20 0.44
LMNA P02545 2/20 0.44
HPGD P15428 2/20 0.44
MTOR P42345 1/20 0.44
METAP2 P50579 1/20 0.44
METAP1 P53582 1/20 0.44
ALDH1A1 P00352 3/20 0.42
NPSR1 Q6W5P4 2/20 0.42
KDM4E B2RXH2 1/20 0.42
ABCB11 O95342 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Timoprazole SCHEMBL563458 1.00 CYP1A2 (0.51) CYP1A2CYP2E1CYP2C8CYP2D6CYP2C9
Timoprazole SCHEMBL9247237 1.00 CYP1A2 (0.51) CYP1A2CYP2E1CYP2C8CYP2D6CYP2C9
Timoprazole SCHEMBL11245124 0.99 CYP1A2 (0.50) CYP1A2CYP2E1CYP2C8CYP2D6CYP2C9
Timoprazole SCHEMBL9244884 0.99 CYP1A2 (0.50) CYP1A2CYP2E1CYP2C8CYP2D6CYP2C9
SCHEMBL8138606 0.86 CYP1A2 (0.49) CYP1A2CYP2E1CYP2C8CYP2D6CYP2C9
SCHEMBL11373497 0.85 KDM4E (0.48) CYP1A2CYP2E1CYP2C8CYP2D6CYP2C9
SCHEMBL27858001 0.84 METAP1 (0.46) CYP1A2CYP2E1CYP2C8CYP2D6CYP2C9
SCHEMBL6872775 0.84 CBFB (0.51) CYP1A2CYP2E1CYP2C8CYP2D6CYP2C9
SCHEMBL6877256 0.84 ALDH1A1 (0.40) CYP1A2CYP2E1CYP2C8CYP2D6CYP2C9
SCHEMBL6440386 0.84 CBFB (0.40) CYP1A2CYP2E1CYP2C8CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1603 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3965735-A1 PHARMACEUTICAL FORMULATION Alkaloid AD Skopje (MK) 2022-03-16 EP claimed
US-20210205270-A1 DRUG COMPOSITIONS FIRST-CITIZENS BANK & TRUST COMPANY, AS ADMINISTRATIVE AGENT 2021-07-08 US claimed
WO-2020224936-A1 PHARMACEUTICAL FORMULATION ALKALOID AD SKOPJE (MK) 2020-11-12 WO claimed
EP-3720844-A1 DRUG COMPOSITIONS Adamis Pharmaceuticals Corporation (US) 2020-10-14 EP claimed
WO-2019113493-A1 DRUG COMPOSITIONS ADAMIS PHARMACEUTICALS CORPORATION (US) 2019-06-13 WO claimed
US-10130618-B2 Pharmaceutical combinations of dabigatran and proton pump inhibitors SANOVEL ILAC SANAYI VE TICARET ANONIM SIRKETI (TR) 2018-11-20 US claimed
CN-107698515-A A kind of preparation method of benzimidazole complex compound 拉萨泰达医药科技有限公司 2018-02-16 CN claimed
EP-2521531-B1 SKIN LIGHTENING COMPOSITIONS ELC MAN LLC (US) 2017-07-12 EP claimed
US-20170035745-A1 PHARMACEUTICAL COMBINATIONS OF DABIGATRAN AND PROTON PUMP INHIBITORS SANOVEL ILAC SANAYI VE TICARET ANONIM SIRKETI (TR) 2017-02-09 US claimed
US-20170035672-A1 SKIN LIGHTENING COMPOSITIONS ELC MAN LLC (US) 2017-02-09 US claimed
EP-0332647-A1 NEW BENZIMIDAZOLE DERIVATIVES A PROCESS FOR PRODUCTION THEREOF AND A PHARMACEUTICAL COMPOSITION CONTAINING THE SAME Aktiebolaget Hässle (SE) 1989-09-20 EP claimed
EP-0279149-A2 Benzimidazole derivatives, process for their production and a pharmaceutical composition containing the same Aktiebolaget Hässle (SE) 1988-08-24 EP claimed
WO-1988003921-A1 NEW BENZIMIDAZOLE DERIVATIVES A PROCESS FOR PRODUCTION THEREOF AND A PHARMACEUTICAL COMPOSITION CONTAINING THE SAME Aktiebolaget Hässle (SE) 1988-06-02 WO claimed
EP-0045200-B1 BENZIMIDAZOLES AND THEIR PHARMACEUTICAL USE THE UPJOHN COMPANY (US) 1988-03-02 EP claimed
EP-0233284-A1 PHARMACOLOGICAL COMPOUNDS. HAESSLE AB (SE) 1987-08-26 EP claimed
WO-1987002668-A1 NOVEL PHARMACOLOGICAL COMPOUNDS Aktiebolaget Hässle (SE) 1987-05-07 WO claimed
EP-0221041-A2 Benzimidazole derivatives, process for their preparation and their pharmaceutical use Aktiebolaget Hässle (SE) 1987-05-06 EP claimed
US-4359465-A HETEROCYCLIC ALKYLSULFINYL BENZIMIDAZOLES THE UPJOHN COMPANY (US) 1982-11-16 US claimed
EP-0045200-A1 Benzimidazoles and their pharmaceutical use THE UPJOHN COMPANY (US) 1982-02-03 EP claimed
US-4045563-A Substituted 2-[pyridylalkylenesulfinyl]-benzimidazoles with gastric acid secretion inhibiting effects AB HASSLE (SW) 1977-08-30 US claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20170035745-A1 PHARMACEUTICAL COMBINATIONS OF DABIGATRAN AND PROTON PUMP INHIBITORS ABCB11, SLC9A5, SLC9A3 CYP1A2 216/4885CYP2E1 454/4885CYP2C8 308/4885
US-20170035672-A1 SKIN LIGHTENING COMPOSITIONS CUTA, TYR, DSG1 CYP1A2 1093/4885CYP2E1 2659/4885CYP2C8 3954/4885
US-10130618-B2 Pharmaceutical combinations of dabigatran and proton pump inhibitors ABCB11, SLC9A5, SLC9A3 CYP1A2 216/4885CYP2E1 454/4885CYP2C8 308/4885
US-20210205270-A1 DRUG COMPOSITIONS CYP2C19, CYP2D6, CYP2B6 CYP1A2 23/4885CYP2E1 19/4885CYP2C8 11/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.