SCHEMBL4649992

SCHEMBL4649992

O=C(O)c1c[nH]c2cc(Cl)c(Cc3ccc(Br)cc3F)cc2c1=O

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.47
ALDH1A1 P00352 2/20 0.42
HPGD P15428 2/20 0.42
MEN1 O00255 1/20 0.42
CYP1A2 P05177 1/20 0.42
ALOX12 P18054 1/20 0.42
KMT2A Q03164 1/20 0.42
GABRA1 P14867 1/20 0.42
GABRB1 P18505 1/20 0.42
GABRA3 P34903 1/20 0.42
GABRB2 P47870 1/20 0.42
MDH2 P40926 2/20 0.41
PRKAB2 O43741 6/20 0.41
PRKAG1 P54619 6/20 0.41
PRKAA2 P54646 6/20 0.41
PRKAA1 Q13131 6/20 0.41
PRKAG3 Q9UGI9 6/20 0.41
PRKAG2 Q9UGJ0 6/20 0.41
PRKAB1 Q9Y478 6/20 0.41
SMN1; SMN2 Q16637 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4650145 0.89 KDM4E (0.51) KDM4EALDH1A1HPGDMEN1CYP1A2
SCHEMBL4650048 0.81 KDM4E (0.50) KDM4EALDH1A1HPGDMEN1CYP1A2
SCHEMBL4650034 0.81 KDM4E (0.49) KDM4EALDH1A1HPGDMEN1CYP1A2
SCHEMBL4649270 0.80 KDM4E (0.57) KDM4EALDH1A1HPGDMEN1CYP1A2
SCHEMBL6713044 0.79 MDH2 (0.55) KDM4EALDH1A1HPGDGABRA1GABRB1
SCHEMBL6714522 0.76 HTT (0.51) KDM4EALDH1A1HPGDMEN1CYP1A2
SCHEMBL10478126 0.76 KDM4E (0.60) KDM4EALDH1A1HPGDMEN1CYP1A2
SCHEMBL6717561 0.76 MDH2 (0.54) KDM4EALDH1A1HPGDGABRA1GABRB1
SCHEMBL4650115 0.76 KDM4E (0.41) KDM4EALDH1A1HPGDMEN1CYP1A2
SCHEMBL4650661 0.75 ALDH1A1 (0.60) KDM4EALDH1A1HPGDMEN1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1963271-A1 QUINOLONE M1 RECEPTOR POSITIVE ALLOSTERIC MODULATORS Merck & Co., Inc. (US) 2008-09-03 EP disclosed
WO-2007067489-A1 QUINOLONE M1 RECEPTOR POSITIVE ALLOSTERIC MODULATORS MERCK & CO., INC. (US) 2007-06-14 WO disclosed