SCHEMBL4650129

SCHEMBL4650129

O=C(O)c1c[nH]c2c(Cc3ccc(OC(F)(F)F)cc3)c(Cl)c(F)cc2c1=O

nearest known ligand 0.43

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CSNK2A2 P19784 3/20 0.42
CSNK2B P67870 3/20 0.42
CSNK2A1 P68400 3/20 0.42
MDH2 P40926 2/20 0.41
AKR1C2 P52895 1/20 0.38
AKR1C1 Q04828 1/20 0.38
ALDH1A1 P00352 3/20 0.38
HPGD P15428 3/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
HAT1 O14929 1/20 0.37
EP300 Q09472 1/20 0.37
MEN1 O00255 1/20 0.37
CYP1A2 P05177 1/20 0.37
ALOX12 P18054 1/20 0.37
KMT2A Q03164 1/20 0.37
KDM4E B2RXH2 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4649429 0.87 ALDH1A1 (0.49) CSNK2A2CSNK2BCSNK2A1ALDH1A1HPGD
SCHEMBL4650054 0.87 CSNK2A2 (0.48) CSNK2A2CSNK2BCSNK2A1MDH2ALDH1A1
SCHEMBL17769720 0.85 CSNK2A2 (0.49) CSNK2A2CSNK2BCSNK2A1MDH2ALDH1A1
SCHEMBL4649277 0.84 ALDH1A1 (0.41) MDH2ALDH1A1HPGDSMN1; SMN2HAT1
SCHEMBL4650001 0.77 CSNK2A2 (0.39) CSNK2A2CSNK2BCSNK2A1MDH2AKR1C2
SCHEMBL5194351 0.76 CSNK2A2 (0.50) CSNK2A2CSNK2BCSNK2A1ALDH1A1HPGD
SCHEMBL4649431 0.76 MDH2 (0.52) MDH2ALDH1A1HPGDSMN1; SMN2MEN1
SCHEMBL4650158 0.76 GABRA1 (0.58) MDH2ALDH1A1HPGDSMN1; SMN2KDM4E
SCHEMBL3812191 0.75 CSNK2A2 (0.49) CSNK2A2CSNK2BCSNK2A1ALDH1A1HPGD
SCHEMBL4650110 0.75 KDM5A (0.42) MDH2ALDH1A1HPGDSMN1; SMN2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1963271-A1 QUINOLONE M1 RECEPTOR POSITIVE ALLOSTERIC MODULATORS Merck & Co., Inc. (US) 2008-09-03 EP claimed
WO-2007067489-A1 QUINOLONE M1 RECEPTOR POSITIVE ALLOSTERIC MODULATORS MERCK & CO., INC. (US) 2007-06-14 WO claimed