SCHEMBL4650265

SCHEMBL4650265

Clc1ccccc1-c1ccc(CN2CCNCC2)c(-c2ccccc2)c1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 3/20 0.48
PDCD1 Q15116 1/20 0.45
CD274 Q9NZQ7 1/20 0.45
LMNA P02545 2/20 0.45
CYP1A2 P05177 1/20 0.45
CYP3A4 P08684 1/20 0.45
CYP2C19 P33261 1/20 0.45
CLK4 Q9HAZ1 1/20 0.45
HTR7 P34969 4/20 0.44
CYP2A6 P11509 1/20 0.44
PTPN11 Q06124 1/20 0.42
DRD2 P14416 1/20 0.42
DRD4 P21917 1/20 0.42
DRD3 P35462 1/20 0.42
MLNR O43193 1/20 0.41
HTR1A P08908 1/20 0.41
HTR2A P28223 1/20 0.41
HTR5A P47898 1/20 0.41
HTR6 P50406 1/20 0.41
MAPK14 Q16539 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27966164 0.82 SIGMAR1 (0.62) SIGMAR1MLNRMAPK14CNR2CXCR4
SCHEMBL7102078 0.81 LMNA (0.55) SIGMAR1LMNAHTR7PTPN11MAPK14
SCHEMBL2472212 0.80 HTR7 (0.64) SIGMAR1LMNAHTR7DRD2DRD4
SCHEMBL30616744 0.80 HTR7 (0.64) SIGMAR1LMNAHTR7DRD2DRD4
SCHEMBL7097670 0.80 LMNA (0.49) SIGMAR1PDCD1CD274LMNAHTR7
SCHEMBL376781 0.78 HTR7 (0.56) SIGMAR1LMNAHTR7MLNRCXCR4
SCHEMBL7098972 0.77 HTR7 (0.59) SIGMAR1PDCD1CD274LMNACYP1A2
Hydrochloric Acid SCHEMBL5689236 0.77 HTR7 (0.55) SIGMAR1LMNAHTR7MLNRCXCR4
Hydrochloric Acid SCHEMBL30688262 0.77 HTR7 (0.55) SIGMAR1LMNAHTR7MLNRCXCR4
Acetic Acid SCHEMBL11195900 0.75 LMNA (0.50) SIGMAR1LMNACYP1A2CYP3A4CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1902014-A2 GLUTAMATE AGGRECANASE INHIBITORS Wyeth (US) 2008-03-26 EP claimed
WO-2007008994-A2 GLUTAMATE AGGRECANASE INHIBITORS WYETH (US) 2007-01-18 WO claimed