SCHEMBL4650433

SCHEMBL4650433

NC(=O)c1ccc(F)cc1-c1ccc(Cl)c(F)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CASP1 P29466 1/20 0.42
ALOX5AP P20292 1/20 0.40
FEN1 P39748 1/20 0.40
KMO O15229 2/20 0.40
CES2 O00748 1/20 0.40
CES1 P23141 1/20 0.40
KMT2A Q03164 2/20 0.39
KDM4E B2RXH2 1/20 0.39
MEN1 O00255 1/20 0.39
USP2 O75604 1/20 0.39
ALDH1A1 P00352 1/20 0.39
DHFR P00374 1/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
LMNA P02545 1/20 0.39
TTR P02766 1/20 0.39
ALB P02768 1/20 0.39
HMGB1 P09429 1/20 0.39
HPGD P15428 1/20 0.39
CXCL12 P48061 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2934440 0.89 EIF4E (0.44) CASP1KMT2ACHRM3ATMMKNK1
SCHEMBL5616409 0.88 CASP1 (0.55) CASP1KMT2AMEN1ALDH1A1CHRM3
SCHEMBL22320212 0.86 IDO1 (0.44) CASP1ALOX5APFEN1CES2CES1
SCHEMBL3904946 0.83 ALOX5AP (0.56) CASP1ALOX5APFEN1KMOKMT2A
SCHEMBL5616523 0.83 CASP1 (0.46) CASP1KDM4EALDH1A1MAPK14IKBKB
SCHEMBL5616614 0.82 IKBKB (0.51) CES2CES1KMT2AMEN1DGAT1
SCHEMBL4650415 0.82 AKR1C3 (0.45) ALOX5APFEN1KMOCES2CES1
SCHEMBL20573272 0.78 BCL9 (0.44) KMOCHRM3
SCHEMBL28142061 0.78 IKBKB (0.48) CES2CES1KMT2AMEN1DGAT1
SCHEMBL4615110 0.77 EIF4E (0.47) CASP1EIF4EPDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1856054-B1 PYRAZOLYLCARBOXANILIDES BAYER CROPSCIENCE AG (DE) 2008-09-17 EP disclosed
EP-1856054-A1 PYRAZOLYLCARBOXANILIDES Bayer CropScience AG (DE) 2007-11-21 EP disclosed
WO-2006092213-A1 PYRAZOLYLCARBOXANILIDES BAYER CROPSCIENCE AG (DE) 2006-09-08 WO disclosed