SCHEMBL4654909

SCHEMBL4654909

CC(=O)Nc1cccc(-c2ccc(N)cc2)c1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.67
CYP17A1 P05093 2/20 0.59
CYP11B1 P15538 1/20 0.59
CYP11B2 P19099 1/20 0.59
MAP4K4 O95819 1/20 0.59
HSD17B1 P14061 1/20 0.58
HSD17B2 P37059 1/20 0.58
MEN1 O00255 1/20 0.57
KMT2A Q03164 1/20 0.57
FYN P06241 1/20 0.56
USP7 Q93009 1/20 0.56
NQO2 P16083 2/20 0.56
PIP4K2A P48426 1/20 0.54
PIP4K2B P78356 1/20 0.54
MGLL Q99685 1/20 0.54
CYP1A2 P05177 1/20 0.54
HSD17B10 Q99714 1/20 0.54
CHEK2 O96017 1/20 0.54
HDAC3 O15379 1/20 0.54
HDAC1 Q13547 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6798003 0.88 ALDH1A1 (0.80) ALDH1A1CYP17A1CYP11B1CYP11B2MAP4K4
SCHEMBL8577619 0.88 SMN1; SMN2 (0.70) ALDH1A1CYP17A1CYP11B1CYP11B2HSD17B1
SCHEMBL3786463 0.86 NQO2 (0.73) ALDH1A1CYP17A1CYP11B1CYP11B2HSD17B1
SCHEMBL12999591 0.85 NPC1 (0.69) ALDH1A1CYP17A1CYP11B1CYP11B2MAP4K4
SCHEMBL12919978 0.84 CYP17A1 (0.60) ALDH1A1CYP17A1CYP11B1CYP11B2HSD17B1
SCHEMBL14384612 0.83 CNR1 (0.71) CYP17A1CYP11B1CYP11B2HSD17B1HSD17B2
SCHEMBL969807 0.83 RAB9A (0.65) ALDH1A1CYP17A1CYP11B1CYP11B2MAP4K4
SCHEMBL6796771 0.83 ALDH1A1 (0.67) ALDH1A1CYP17A1CYP11B1CYP11B2MAP4K4
SCHEMBL1016291 0.83 ALDH1A1 (0.57) ALDH1A1CYP17A1CYP11B1CYP11B2MAP4K4
SCHEMBL3225408 0.82 SMN1; SMN2 (0.79) ALDH1A1MEN1KMT2AHSD17B10HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1976842-B1 MODULATORS OF ALPHA7 NICOTINIC ACETYLCHOLINE RECEPTORS AND THERAPEUTIC USES THEREOF SIENA BIOTECH SPA (IT) 2010-03-10 EP disclosed
EP-1991528-A2 MODULATORS OF ALPHA7 NICOTINIC ACETYLCHOLINE RECEPTORS AND THERAPEUTIC USES THEREOF Siena Biotech S.p.A. (IT) 2008-11-19 EP disclosed
WO-2007098826-A2 MODULATORS OF ALPHA7 NICOTINIC ACETYLCHOLINE RECEPTORS AND THERAPEUTIC USES THEREOF SIENA BIOTECH S.P.A. (IT) 2007-09-07 WO disclosed