SCHEMBL4656709

SCHEMBL4656709

CCCCCOc1ccc(NC(N)=O)cc1F

nearest known ligand 0.64

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MAPT P10636 1/20 0.64
HSD17B10 Q99714 1/20 0.64
S1PR1 P21453 4/20 0.60
S1PR3 Q99500 2/20 0.60
S1PR4 O95977 1/20 0.60
S1PR5 Q9H228 1/20 0.60
THRA P10827 1/20 0.50
THRB P10828 1/20 0.50
C5 P01031 1/20 0.47
S1PR2 O95136 1/20 0.46
LPAR2 Q9HBW0 1/20 0.46
FAAH O00519 7/20 0.46
STS P08842 1/20 0.46
ALDH1A1 P00352 1/20 0.46
SMPD1 P17405 3/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9885402 0.88 S1PR1 (0.58) MAPTHSD17B10S1PR1S1PR3S1PR4
SCHEMBL13338000 0.86 S1PR1 (0.54) MAPTHSD17B10S1PR1S1PR3S1PR4
SCHEMBL26554065 0.84 S1PR1 (0.58) S1PR1S1PR3S1PR4S1PR5THRA
SCHEMBL12164847 0.81 S1PR4 (0.52) MAPTHSD17B10S1PR1S1PR3S1PR4
SCHEMBL28203083 0.79 S1PR1 (0.51) S1PR1S1PR3S1PR4S1PR5THRA
SCHEMBL4401762 0.78 MAPT (0.57) MAPTHSD17B10S1PR1S1PR3S1PR4
SCHEMBL6512897 0.77 MAPK1 (0.59) MAPTALDH1A1
SCHEMBL9440250 0.76 THRA (0.67) S1PR1S1PR3S1PR4S1PR5THRA
SCHEMBL23554170 0.76 ALDH1A1 (0.69) S1PR1S1PR3FAAHALDH1A1
SCHEMBL9503837 0.76 ALDH1A1 (0.69) S1PR1S1PR3FAAHALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1996565-A2 SUBSTITUTED AMINOTHIAZOLE DERIVATIVES WITH ANTI-HCV ACTIVITY Achillion Pharmaceuticals, Inc. (US) 2008-12-03 EP disclosed
WO-2007103550-A2 SUBSTITUTED AMINOTHIAZOLE DERIVATIVES WITH ANTI-HCV ACTIVITY ACHILLION PHARMACEUTICALS, INC. (US) 2007-09-13 WO disclosed